# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | SR-318 | 93; SR-318 | IC50 | = | 14 | uM | ALA5213217 | 4.85 | nM | Homo sapiens | ||
2. | SR-318 | 93; SR-318 | % of control | = | 29 | % | ALA5213216 | % | Homo sapiens | |||
3. | ALA4518706 | EUB0000702 | % of control | = | 4.6 | % | ALA5213300 | % | Homo sapiens | |||
4. | Enzastaurin (LY317615) | 1e | Kd | = | 25 | nM | ALA5214801 | 7.60 | nM | Homo sapiens | ||
5. | BAY-985 | 34; BAY-985 | IC50 | = | 276 | nM | ALA5213259 | 6.56 | nM | Homo sapiens | ||
6. | GSK461364 | GSK-461364A | % of inhibition | = | 92 | % | ALA5214848 | % | Homo sapiens | |||
7. | GSK2334470 | (3S,6R)-28d, GSK-2334470 | % of control | = | 12 | % | ALA5212811 | % | Homo sapiens | |||
8. | FM-381 | FM-381 | % of inhibition | = | 60 | % | ALA5213570 | % | Homo sapiens | |||
9. | ALA4531220 | EUB0000586 | % of control | = | 0 | % | ALA5214754 | % | Homo sapiens | |||
10. | ALA4445335 | Roxyl-ZV-5J | INH | = | 22 | % | ALA4408125 | % | Homo sapiens | |||
11. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405558 | % | Homo sapiens | |||
12. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405557 | % | Homo sapiens | |||
13. | ALA4559936 | (+/-)-6 | Activity | = | 57 | % | ALA4391579 | % | Homo sapiens | |||
14. | ALA4559936 | (+/-)-6 | Activity | = | 2.2 | % | ALA4391578 | % | Homo sapiens | |||
15. | ALA4564973 | 50 | INH | = | 88 | % | ALA4389953 | % | Homo sapiens | |||
16. | ALA4564973 | 50 | INH | = | 89 | % | ALA4389952 | % | Homo sapiens | |||
17. | ALA4555459 | 43 | INH | = | 34 | % | ALA4389475 | % | Homo sapiens | |||
18. | ALA4555459 | 43 | INH | = | 50 | % | ALA4389476 | % | Homo sapiens | |||
19. | ALA4473365 | 7c | Activity | = | 15 | % | ALA4382757 | % | Homo sapiens | |||
20. | ALA4473365 | 7c | Activity | = | 15 | % | ALA4382756 | % | Homo sapiens |