| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Cannabidiol | 3 | Ki | = | 12.3 | uM | ALA4687736 | 4.91 | nM | Homo sapiens | ||
| 2. |  ALA4203313 | 12 | Drug metabolism | 0 | ALA4185366 | Metabolite_Notdetected | Homo sapiens | |||||
| 3. |  rac 6-Chloro-1,4-dihydro-4-(1-pentynyl)-4-(trifluoromethyl)-2H-3,1-benzoxazin-2-one | 4 | Drug metabolism | 0 | ALA3388988 | metabolite_detected | Homo sapiens | |||||
| 4. |  ALA3344473 | 3 | Drug metabolism | 0 | ALA3388988 | metabolite_detected | Homo sapiens | |||||
| 5. |  Budesonide | Budesonide(2) | Drug metabolism | 0 | ALA3541872 | metabolite_detected | Homo sapiens | |||||
| 6. | Budesonide | Budesonide(2) | Drug metabolism | 0 | ALA3541869 | metabolite_detected | Homo sapiens | |||||
| 7. |  ALA3526818 | [14C]-Fingolimod, FTY720 | Drug metabolism | 0 | ALA3533014 | metabolite_not_detected | Homo sapiens | |||||
| 8. |  ALA3527325 | M3 | Vmax | = | 0.286 | nmol/min | ALA3538281 | nmol/min | Homo sapiens | |||
| 9. | ALA3527325 | M3 | Km | = | 37.4 | uM | ALA3538281 | nM | Homo sapiens | |||
| 10. |  ALA3527324 | M2 | Vmax | = | 0.26 | nmol/min | ALA3538281 | nmol/min | Homo sapiens | |||
| 11. | ALA3527324 | M2 | Km | = | 10 | uM | ALA3538281 | nM | Homo sapiens | |||
| 12. |  AMG 853 | 5, AMG-853 | Drug metabolism | 0 | ALA3538085 | metabolite_detected | Homo sapiens | |||||
| 13. | ALA3527325 | M3 | Drug metabolism | 0 | ALA3537749 | metabolite_detected | Homo sapiens | |||||
| 14. | ALA3527324 | M2 | Drug metabolism | 0 | ALA3537749 | metabolite_detected | Homo sapiens | |||||
| 15. | AMG 853 | 5, AMG-853 | Drug metabolism | 0 | ALA3537744 | metabolite_detected | Homo sapiens | |||||
| 16. |  ALA3542193 | 23-hydroxy budesonide | Drug metabolism | 0 | ALA3539426 | metabolite_detected | Homo sapiens | |||||
| 17. |  6β-Hydroxy Budesonide | 6beta-hydroxy budesonide | Drug metabolism | 0 | ALA3539426 | metabolite_detected | Homo sapiens | |||||
| 18. |  PF-4981517 | CYP3cide, PF-04981517 | INH | = | 15 | % | ALA3532546 | % | Homo sapiens | |||
| 19. | PF-4981517 | CYP3cide, PF-04981517 | IC50 | = | 33 | uM | ALA3532654 | 4.48 | nM | Homo sapiens | ||
| 20. | Budesonide | Budesonide(2) | Drug metabolism | 0 | ALA3539729 | metabolite_not_detected | Homo sapiens |
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