# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3335388 | YAP(81-100) | INH | = | 60 | % | ALA3385959 | % | Homo sapiens | |||
2. | ALA3335391 | YAP(84-100) | INH | = | 62 | % | ALA3385959 | % | Homo sapiens | |||
3. | ALA3335394 | YAP(87-100) | INH | = | 12 | % | ALA3385959 | % | Homo sapiens | |||
4. | ALA3335397 | YAP(81-97) | INH | = | 14 | % | ALA3385959 | % | Homo sapiens | |||
5. | ALA3335400 | YAP(T83A) | INH | = | 52 | % | ALA3385959 | % | Homo sapiens | |||
6. | ALA3335430 | YAP(M86A) | INH | = | 1.3 | % | ALA3385959 | % | Homo sapiens | |||
7. | ALA3335433 | YAP(R89A) | INH | = | 1.7 | % | ALA3385959 | % | Homo sapiens | |||
8. | ALA3335436 | YAP(P92A) | INH | = | 0 | % | ALA3385959 | % | Homo sapiens | |||
9. | ALA3335439 | YAP(F95A) | INH | = | 4 | % | ALA3385959 | % | Homo sapiens | |||
10. | ALA3335442 | YAP(P98A) | INH | = | 47 | % | ALA3385959 | % | Homo sapiens | |||
11. | ALA3335388 | YAP(81-100) | IC50 | = | 49 | uM | ALA3385960 | 4.31 | nM | Homo sapiens | ||
12. | ALA3335444 | YAP(E100A) | IC50 | = | 43 | uM | ALA3385960 | 4.37 | nM | Homo sapiens | ||
13. | ALA3335447 | 3 | IC50 | = | 6.9 | uM | ALA3385960 | 5.16 | nM | Homo sapiens | ||
14. | ALA3335450 | 6 | IC50 | = | 1.5 | uM | ALA3385960 | 5.82 | nM | Homo sapiens | ||
15. | ALA3335453 | 9 | IC50 | = | 0.042 | uM | ALA3385960 | 7.38 | nM | Homo sapiens | ||
16. | ALA3335456 | 12 | IC50 | = | 0.31 | uM | ALA3385960 | 6.51 | nM | Homo sapiens | ||
17. | ALA3335459 | 15 | IC50 | = | 0.35 | uM | ALA3385960 | 6.46 | nM | Homo sapiens | ||
18. | ALA3335462 | 18 | IC50 | = | 0.53 | uM | ALA3385960 | 6.28 | nM | Homo sapiens | ||
19. | ALA3335452 | 8 | Kd | = | 39 | nM | ALA3385961 | 7.41 | nM | Homo sapiens | ||
20. | ALA3335389 | YAP(82-100) | INH | = | 59 | % | ALA3385959 | % | Homo sapiens |