# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Drug uptake | 0 | ALA3541985 | Active | Bos taurus | |||||
2. | [³H]taurocholic acid | THCA | Drug uptake | 0 | ALA3541986 | Active | Bos taurus | |||||
3. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Drug uptake | 0 | ALA3541987 | Active | Bos taurus | |||||
4. | [³H]taurocholic acid | THCA | Drug uptake | 0 | ALA3541988 | Active | Bos taurus | |||||
5. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Km | = | 0.25 | uM | ALA3538497 | nM | Bos taurus | |||
6. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Km | = | 46.6 | uM | ALA3538498 | nM | Bos taurus | |||
7. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Vmax | = | 24.5 | pmol/mg/min | ALA3538497 | pmol/mg/min | Bos taurus | |||
8. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Vmax | = | 375 | pmol/mg/min | ALA3538498 | pmol/mg/min | Bos taurus | |||
9. | [³H]taurocholic acid | THCA | Km | = | 40.2 | uM | ALA3538500 | nM | Bos taurus | |||
10. | [³H]taurocholic acid | THCA | Vmax | = | 55.4 | pmol/mg/min | ALA3538500 | pmol/mg/min | Bos taurus | |||
11. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Drug uptake | 0 | ALA3538501 | Active | Bos taurus | |||||
12. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Drug uptake | 0 | ALA3538502 | Active | Bos taurus | |||||
13. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Drug uptake | 0 | ALA3538503 | Active | Bos taurus | |||||
14. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Drug uptake | 0 | ALA3538504 | Active | Bos taurus | |||||
15. | [³H]taurocholic acid | THCA | Drug uptake | 0 | ALA3538505 | Active | Bos taurus | |||||
16. | [³H]taurocholic acid | THCA | Drug uptake | 0 | ALA3538506 | Active | Bos taurus | |||||
17. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Drug uptake | 0 | ALA3538507 | Not Active | Bos taurus | |||||
18. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Drug uptake | 0 | ALA3538508 | Active | Bos taurus | |||||
19. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Drug uptake | 0 | ALA3538509 | Not Active | Bos taurus | |||||
20. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Drug uptake | 0 | ALA3538510 | Not Active | Bos taurus |