# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3403619 | 22b, enantiomer-2 | Emax | = | 82 | % | ALA3404961 | % | Macaca mulatta | |||
2. | ALA3359523 | 25 | Emax | = | 84 | % | ALA3380164 | % | Macaca mulatta | |||
3. | ALA3359522 | 24 | Emax | = | 96 | % | ALA3380164 | % | Macaca mulatta | |||
4. | ALA3359523 | 25 | EC50 | = | 0.058 | nM | ALA3380163 | 10.24 | nM | Macaca mulatta | ||
5. | ALA3359522 | 24 | EC50 | = | 0.038 | nM | ALA3380163 | 10.42 | nM | Macaca mulatta | ||
6. | etrasimod | (R)-4, APD334 | EC50 | = | 0.32 | nM | ALA3380996 | 9.49 | nM | Macaca mulatta | ||
7. | etrasimod | (R)-4, APD334 | Emax | = | 95 | % | ALA3380997 | % | Macaca mulatta |