# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3408356 | Lac-ENF | Kd | = | 452 | nM | ALA3412776 | 6.34 | nM | Human immunodeficiency virus 1 | ||
2. | Enfuvirtide | DP178 | Kd | = | 182 | nM | ALA3412776 | 6.74 | nM | Human immunodeficiency virus 1 | ||
3. | ALA3408357 | SL-ENF | Kd | = | 250 | nM | ALA3412776 | 6.60 | nM | Human immunodeficiency virus 1 | ||
4. | Enfuvirtide | DP178 | Activity | = | 67 | % | ALA3412777 | % | Human immunodeficiency virus 1 | |||
5. | ALA3408356 | Lac-ENF | Activity | = | 118 | % | ALA3412777 | % | Human immunodeficiency virus 1 | |||
6. | ALA3408357 | SL-ENF | Activity | = | 157 | % | ALA3412777 | % | Human immunodeficiency virus 1 | |||
7. | NBD-556 | NBD-556 | IC50 | = | 0.61 | uM | ALA3385405 | 6.21 | nM | Human immunodeficiency virus 1 | ||
8. | ALA2380932 | C34 | INH | 0 | ALA3366759 | Active | % | Human immunodeficiency virus 1 | ||||
9. | ALA3341854 | P26-BApc | INH | 0 | ALA3366759 | Active | % | Human immunodeficiency virus 1 | ||||
10. | ALA2380932 | C34 | IC50 | = | 2.84 | uM | ALA3366758 | 5.55 | nM | Human immunodeficiency virus 1 | ||
11. | ALA3341859 | Ptrz-P26 | INH | 0 | ALA3366758 | Not Active | % | Human immunodeficiency virus 1 | ||||
12. | ALA3341857 | P26-OApc | IC50 | = | 8.31 | uM | ALA3366758 | 5.08 | nM | Human immunodeficiency virus 1 | ||
13. | ALA3341856 | P26-UApc | IC50 | = | 8.31 | uM | ALA3366758 | 5.08 | nM | Human immunodeficiency virus 1 | ||
14. | ALA3341855 | P26-BApo | IC50 | = | 8.31 | uM | ALA3366758 | 5.08 | nM | Human immunodeficiency virus 1 | ||
15. | ALA3341854 | P26-BApc | IC50 | = | 8.31 | uM | ALA3366758 | 5.08 | nM | Human immunodeficiency virus 1 | ||
16. | ALA3341853 | P26-BAc | IC50 | = | 8.31 | uM | ALA3366758 | 5.08 | nM | Human immunodeficiency virus 1 | ||
17. | ALA3341852 | P26-BAo | IC50 | = | 8.31 | uM | ALA3366758 | 5.08 | nM | Human immunodeficiency virus 1 | ||
18. | ALA2380932 | C34 | Ratio EC50 | > | 769 | ALA3366757 | Human immunodeficiency virus 1 | |||||
19. | Enfuvirtide | DP178 | Ratio EC50 | = | 39 | ALA3366757 | Human immunodeficiency virus 1 | |||||
20. | ALA3341854 | P26-BApc | Ratio EC50 | = | 11 | ALA3366757 | Human immunodeficiency virus 1 |