# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Sunitinib | 12b | IC50 | = | 0.015 | uM | ALA5252745 | 7.82 | nM | Homo sapiens | ||
2. | MnTMPyP pentachloride | 5 | IC50 | = | 0.402 | uM | ALA5252745 | 6.40 | nM | Homo sapiens | ||
3. | AAL 993 | 5 | IC50 | = | 0.13 | uM | ALA5252745 | 6.89 | nM | Homo sapiens | ||
4. | Vatalanib succinate | CGP-79787D | IC50 | = | 0.077 | uM | ALA5252745 | 7.11 | nM | Homo sapiens | ||
5. | ALA5280119 | 10 | IC50 | = | 0.333 | uM | ALA5252745 | 6.48 | nM | Homo sapiens | ||
6. | ALA5276611 | 4 | IC50 | = | 0.223 | uM | ALA5252745 | 6.65 | nM | Homo sapiens | ||
7. | BFH772 | 1 | IC50 | = | 1.7 | uM | ALA5252745 | 5.77 | nM | Homo sapiens | ||
8. | ALA5288744 | 9 | IC50 | = | 0.081 | uM | ALA5252745 | 7.09 | nM | Homo sapiens | ||
9. | BAW2881(NVP-BAW2881) | 2 | IC50 | = | 0.82 | uM | ALA5252745 | 6.09 | nM | Homo sapiens | ||
10. | Staurosporine | 1 (Staurosporine) | Kd | = | 11 | nM | ALA5252319 | 7.96 | nM | Homo sapiens | ||
11. | ALA5271697 | 8a | INH | = | 36 | % | ALA5252308 | % | Homo sapiens | |||
12. | ALA5271697 | 8a | deltaTm | = | 4.2 | degrees C | ALA5252297 | degrees C | Homo sapiens | |||
13. | ALA5274338 | 2e | INH | < | 50 | % | ALA5251045 | % | Homo sapiens | |||
14. | ALA2220486 | LUCITANIB | IC50 | = | 7 | nM | ALA5241426 | 8.15 | nM | Homo sapiens | ||
15. | ALA522892 | 5 | IC50 | = | 8 | nM | ALA5241416 | 8.10 | nM | Homo sapiens | ||
16. | ODM-203 | BDBM247327 | IC50 | = | 26 | nM | ALA5241393 | 7.58 | nM | Homo sapiens | ||
17. | ALA4278642 | 25e; SOMCL-085 | IC50 | = | 5.6 | nM | ALA5241385 | 8.25 | nM | Homo sapiens | ||
18. | GSK1070916 | GSK-1070916 | IC50 | = | 42 | nM | ALA5213115 | 7.38 | nM | Homo sapiens | ||
19. | BAY1125976 | BAY-1125976 | Kd | = | 210 | nM | ALA5213035 | 6.68 | nM | Homo sapiens | ||
20. | ALA3417525 | 69, BI665915 | % of inhibition | = | 64 | % | ALA5214008 | % | Homo sapiens |