# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA334721 | MEN-10627 | pA2 | = | 8.21 | ALA812066 | 8.21 | nM | Rattus norvegicus | |||
2. | ALA334721 | MEN-10627 | Emax | = | 94 | % | ALA814856 | % | Rattus norvegicus | |||
3. | ALA334721 | MEN-10627 | Emax | = | 96 | % | ALA811994 | % | Rattus norvegicus | |||
4. | ALA334721 | MEN-10627 | Emax | = | 95 | % | ALA814857 | % | Rattus norvegicus | |||
5. | L-732,138 | 26 (L) | Ki | = | 134 | nM | ALA1217615 | 6.87 | nM | Rattus norvegicus | ||
6. | L-732,138 | 26 (L) | pIC50 | = | 6.4 | ALA1217615 | 6.40 | nM | Rattus norvegicus | |||
7. | ALA1214027 | 5 | pIC50 | = | 6.98 | ALA1217615 | 6.98 | nM | Rattus norvegicus | |||
8. | ALA1214026 | 4 | pIC50 | = | 6.18 | ALA1217615 | 6.18 | nM | Rattus norvegicus | |||
9. | ALA1214025 | 3 | pIC50 | = | 7.74 | ALA1217615 | 7.74 | nM | Rattus norvegicus | |||
10. | ALA1214024 | 2 | pIC50 | = | 7.38 | ALA1217615 | 7.38 | nM | Rattus norvegicus | |||
11. | ALA507340 | 2 | pIC50 | = | 7.61 | ALA1217615 | 7.61 | nM | Rattus norvegicus | |||
12. | ALA507340 | 2 | Ki | = | 7.3 | nM | ALA1217615 | 8.14 | nM | Rattus norvegicus | ||
13. | ALA1214024 | 2 | Ki | = | 10 | nM | ALA1217615 | 8.00 | nM | Rattus norvegicus | ||
14. | ALA1214025 | 3 | Ki | = | 4.5 | nM | ALA1217615 | 8.35 | nM | Rattus norvegicus | ||
15. | ALA1214026 | 4 | Ki | = | 160 | nM | ALA1217615 | 6.80 | nM | Rattus norvegicus | ||
16. | ALA1214027 | 5 | Ki | = | 26 | nM | ALA1217615 | 7.58 | nM | Rattus norvegicus | ||
17. | ALA217406 | table II | EC50 | = | 64.8 | nM | ALA1037216 | 7.19 | nM | Rattus norvegicus | ||
18. | ALA217406 | table II | EC50 | = | 0.55 | nM | ALA1037222 | 9.26 | nM | Rattus norvegicus | ||
19. | ALA566469 | 16 | Emax | = | 120 | % | ALA1037221 | % | Rattus norvegicus | |||
20. | ALA567108 | 1 | Activity | 0 | ALA1037221 | Not Active | Rattus norvegicus |