| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4579120 | 40; E40 | INH | = | 48.3 | % | ALA4396150 | % | Homo sapiens | |||
| 2. |  ALA4569878 | 4c | IC50 | > | 100 | uM | ALA4393421 | nM | Homo sapiens | |||
| 3. |  ALA4546800 | (R)-4a | IC50 | = | 0.26 | uM | ALA4393426 | 6.58 | nM | Homo sapiens | ||
| 4. |  ALA4567857 | 4b | IC50 | = | 4.1 | uM | ALA4393426 | 5.39 | nM | Homo sapiens | ||
| 5. | ALA4569878 | 4c | IC50 | = | 10.3 | uM | ALA4393426 | 4.99 | nM | Homo sapiens | ||
| 6. |  ALA4437427 | (R)-4c | IC50 | = | 11.8 | uM | ALA4393426 | 4.93 | nM | Homo sapiens | ||
| 7. |  ALA4516772 | (S)-4c | IC50 | = | 13.7 | uM | ALA4393426 | 4.86 | nM | Homo sapiens | ||
| 8. |  ALA4558106 | 4d | IC50 | = | 8.2 | uM | ALA4393426 | 5.09 | nM | Homo sapiens | ||
| 9. |  ALA4471059 | 19 | INH | = | 3.2 | % | ALA4368591 | % | Homo sapiens | |||
| 10. |  ALA4793451 | 4j; MGS0274 | Activity | 0 | ALA4708806 | Not Active | Homo sapiens | |||||
| 11. |  ALA334014 | 3 | Activity | 0 | ALA4708806 | Not Active | Homo sapiens | |||||
| 12. |  Remibrutinib (LOU064) | 25; LOU064 | Activity | 0 | ALA4358664 | Not Active | Homo sapiens | |||||
| 13. |  ALA75478 | 43 | Ki | = | 945 | nM | ALA4322116 | 6.03 | nM | Homo sapiens | ||
| 14. |  ALA4576324 | 24 | Ki | = | 0.3 | nM | ALA4322116 | 9.52 | nM | Homo sapiens | ||
| 15. |  Belzutifan | 2; PT2977 | Activity | 0 | ALA4312681 | Not Active | Homo sapiens | |||||
| 16. |  CHDI 00390576 | 22 | INH | < | 25 | % | ALA4311064 | % | Homo sapiens | |||
| 17. |  ALA4437833 | 16 | INH | < | 25 | % | ALA4311064 | % | Homo sapiens | |||
| 18. |  ALA4202767 | 56 | Activity | <= | 25 | % | ALA4187115 | % | Homo sapiens | |||
| 19. |  ALA4802042 | EUB0001568 | % inhibition | 18 | % | ALA4888408 | Not Active | % | Homo sapiens | |||
| 20. | ALA4802042 | EUB0001568 | % inhibition | 22 | % | ALA4888408 | Not Active | % | Homo sapiens |
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