# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4637208 | EUB0001113 | pKd | 4.5 | ALA4886885 | nM | Homo sapiens | |||||
2. | ALA4637208 | EUB0001113 | pKd | 4.5 | ALA4886884 | nM | Homo sapiens | |||||
3. | GSK620 | 1; 20 | pKd | 4.5 | ALA4885833 | nM | Homo sapiens | |||||
4. | GSK620 | 1; 20 | pKd | 4.5 | ALA4885832 | nM | Homo sapiens | |||||
5. | GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885777 | nM | Homo sapiens | ||||
6. | GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885776 | nM | Homo sapiens | ||||
7. | ALA4648362 | EUB0001116 | pKd | 4.5 | ALA4885709 | nM | Homo sapiens | |||||
8. | ALA4648362 | EUB0001116 | pKd | 4.5 | ALA4885708 | nM | Homo sapiens | |||||
9. | bromosporine | Bromosporine | Delta TM | = | 2.58 | C | ALA4650093 | C | Homo sapiens | |||
10. | ALA4852928 | 60; GSK040 | INH | < | 40 | % | ALA4827476 | % | Homo sapiens | |||
11. | ALA4852928 | 60; GSK040 | INH | < | 40 | % | ALA4827475 | % | Homo sapiens | |||
12. | Mivebresib | BDBM220447 | Kd | > | 1 | uM | ALA4020270 | nM | Homo sapiens | |||
13. | ALA3926851 | BDBM249277 | Kd | > | 10000 | nM | ALA4332529 | nM | Homo sapiens | |||
14. | ALA3926851 | BDBM249277 | Kd | = | 5900 | nM | ALA4332528 | 5.23 | nM | Homo sapiens | ||
15. | ALA4637298 | 36; GSK973 | INH | 0 | ALA4622551 | Not Active | % | Homo sapiens | ||||
16. | ALA4637298 | 36; GSK973 | INH | 0 | ALA4622550 | Not Active | % | Homo sapiens | ||||
17. | ALA4648912 | 27; XL-223 | Kd | < | 1 | nM | ALA4612499 | nM | Homo sapiens | |||
18. | ALA4648912 | 27; XL-223 | Kd | < | 1 | nM | ALA4612498 | nM | Homo sapiens | |||
19. | ALA3968533 | 59 | IC50 | > | 20 | uM | ALA3864409 | nM | Homo sapiens | |||
20. | ALA3959584 | 7 | IC50 | > | 20 | uM | ALA3864409 | nM | Homo sapiens |