| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1472 | TRH | EC50 | = | 0.001 | uM | ALA3602665 | 9.28 | nM | Mus musculus | ||
| 2. |  ALA3600450 | 12e, (2S)-Pip-L-His(2-isopropyl)-L-ProNH2 | EC50 | = | 0.77 | uM | ALA3602665 | 6.11 | nM | Mus musculus | ||
| 3. |  ALA3600449 | 12d, (2S)-Pip-L-His(2-propyl)-L-ProNH2 | EC50 | = | 0.004 | uM | ALA3602665 | 8.40 | nM | Mus musculus | ||
| 4. |  ALA3600448 | 12c, 3-Apyz-L-His(2-propyl)-L-ProNH2 | EC50 | = | 0.12 | uM | ALA3602665 | 6.92 | nM | Mus musculus | ||
| 5. |  ALA3600447 | 12b, 5-Mpyz-L-His(2-propyl)-L-ProNH2 | EC50 | = | 0.015 | uM | ALA3602665 | 7.82 | nM | Mus musculus | ||
| 6. |  ALA3600446 | 12a, 2-Pyz-L-His(2-propyl)-L-ProNH2 | EC50 | = | 0.06 | uM | ALA3602665 | 7.22 | nM | Mus musculus | ||
| 7. |  ALA3600445 | 8l, 2-Pyz-L-His(2,5-diiodo-1-benzyl)-L-ProNH2 | EC50 | = | 0.03 | uM | ALA3602665 | 7.52 | nM | Mus musculus | ||
| 8. |  ALA3600444 | 8k, 5-Mpyz-L-His(2,5-diiodo-1-benzyl)-L-ProNH2 | EC50 | = | 0.05 | uM | ALA3602665 | 7.30 | nM | Mus musculus | ||
| 9. |  ALA3601786 | 8j, 2-Pyz-L-His(2,5-diiodo-1-ethyl)-L-ProNH2 | EC50 | = | 0.96 | uM | ALA3602665 | 6.02 | nM | Mus musculus | ||
| 10. |  ALA3601785 | 8i, 2-Pyz-L-His(5-bromo-1-methyl)-L-ProNH2 | EC50 | = | 0.03 | uM | ALA3602665 | 7.52 | nM | Mus musculus | ||
| 11. |  ALA3601784 | 8h, 2-Pyz-L-His(2,5-diiodo)-L-ProNH2 | EC50 | = | 0.31 | uM | ALA3602665 | 6.51 | nM | Mus musculus | ||
| 12. |  ALA3601783 | 8g, 3-Apyz-L-His(2,5-dibromo)-L-ProNH2 | EC50 | = | 0.29 | uM | ALA3602665 | 6.54 | nM | Mus musculus | ||
| 13. |  ALA3601782 | 8f, 3-Apyz-L-His(5-bromo)-L-ProNH2 | EC50 | = | 0.006 | uM | ALA3602665 | 8.22 | nM | Mus musculus | ||
| 14. |  ALA3601781 | 8e, 5-Mpyz-L-His(5-bromo)-L-ProNH2 | EC50 | = | 0.04 | uM | ALA3602665 | 7.40 | nM | Mus musculus | ||
| 15. |  ALA3600454 | 8d, 2-Mpyz-L-His(2,5-dibromo)-L-ProNH2 | EC50 | = | 0.1 | uM | ALA3602665 | 7.00 | nM | Mus musculus | ||
| 16. |  ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | EC50 | = | 0.05 | uM | ALA3602665 | 7.30 | nM | Mus musculus | ||
| 17. |  ALA3600452 | 8b, 2-Pyz-L-His(5-bromo)-L-ProNH2 | EC50 | = | 0.048 | uM | ALA3602665 | 7.32 | nM | Mus musculus | ||
| 18. |  ALA3600451 | 8a, 2-Pyz-L-His(5-chloro)-L-ProNH2 | EC50 | = | 0.53 | uM | ALA3602665 | 6.28 | nM | Mus musculus | ||
| 19. | ALA3600451 | 8a, 2-Pyz-L-His(5-chloro)-L-ProNH2 | IC50 | > | 50 | uM | ALA3602663 | nM | Mus musculus | |||
| 20. | ALA3600452 | 8b, 2-Pyz-L-His(5-bromo)-L-ProNH2 | IC50 | > | 50 | uM | ALA3602663 | nM | Mus musculus |
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