# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4163247 | 2; BVM | t1/2 | <= | 3 | min | ALA4157509 | hr | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
2. | ALA3827379 | 2; BMS-955176 | t1/2 | = | 46 | min | ALA4157509 | hr | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
3. | ALA4163247 | 2; BVM | t1/2 | <= | 3 | min | ALA4157508 | hr | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
4. | ALA3827379 | 2; BMS-955176 | t1/2 | = | 36 | min | ALA4157508 | hr | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
5. | ALA3827379 | 2; BMS-955176 | Kd | = | 98 | nM | ALA4157402 | 7.01 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | ||
6. | ALA4163247 | 2; BVM | Kd | = | 259 | nM | ALA4157401 | 6.59 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | ||
7. | ALA3827379 | 2; BMS-955176 | Kd | = | 33.6 | nM | ALA4157401 | 7.47 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | ||
8. | ALA4163247 | 2; BVM | Kd | = | 49.2 | nM | ALA4157400 | 7.31 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | ||
9. | ALA3827379 | 2; BMS-955176 | Kd | = | 6.5 | nM | ALA4157400 | 8.19 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | ||
10. | ALA4163247 | 2; BVM | Kd | = | 15 | nM | ALA4157399 | 7.82 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | ||
11. | ALA3827379 | 2; BMS-955176 | Kd | = | 4.3 | nM | ALA4157399 | 8.37 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | ||
12. | Raltegravir (MK-0518) | 1, raltegravir | IC50 | 0 | ALA4135243 | Not Determined | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||||
13. | ALA4163126 | 11m | IC50 | > | 10 | uM | ALA4135243 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
14. | ALA4176527 | 11l | IC50 | > | 10 | uM | ALA4135243 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
15. | ALA4161240 | 11k | IC50 | > | 10 | uM | ALA4135243 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
16. | ALA4168270 | 11j | IC50 | > | 10 | uM | ALA4135243 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
17. | ALA4167025 | 11i | IC50 | > | 10 | uM | ALA4135243 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
18. | ALA4175393 | 11h | IC50 | > | 10 | uM | ALA4135243 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
19. | ALA4170599 | 14 | IC50 | > | 10 | uM | ALA4135243 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
20. | ALA4159305 | 9a | IC50 | > | 10 | uM | ALA4135243 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) |