# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4462110 | (S)-38 | INH | = | 102 | % | ALA4423301 | % | Rattus norvegicus | |||
2. | ALA4532472 | (R)-36 | INH | = | 85 | % | ALA4423301 | % | Rattus norvegicus | |||
3. | ALA4455600 | (S)-33 | INH | = | 103 | % | ALA4423301 | % | Rattus norvegicus | |||
4. | ALA4540313 | (S)-25 | INH | = | 90 | % | ALA4423301 | % | Rattus norvegicus | |||
5. | AZD9977 | BDBM238159 | INH | = | 101 | % | ALA4423301 | % | Rattus norvegicus | |||
6. | ALA4557032 | (S)-11 | INH | = | 103 | % | ALA4423301 | % | Rattus norvegicus | |||
7. | Eplerenone | 1 | INH | = | 102 | % | ALA4423301 | % | Rattus norvegicus | |||
8. | ALA4462110 | (S)-38 | pIC50 | = | 7.1 | ALA4423300 | 7.10 | nM | Rattus norvegicus | |||
9. | ALA4532472 | (R)-36 | pIC50 | = | 8.1 | ALA4423300 | 8.10 | nM | Rattus norvegicus | |||
10. | ALA4455600 | (S)-33 | pIC50 | = | 7 | ALA4423300 | 7.00 | nM | Rattus norvegicus | |||
11. | ALA4540313 | (S)-25 | pIC50 | = | 8 | ALA4423300 | 8.00 | nM | Rattus norvegicus | |||
12. | AZD9977 | BDBM238159 | pIC50 | = | 7.1 | ALA4423300 | 7.10 | nM | Rattus norvegicus | |||
13. | ALA4557032 | (S)-11 | pIC50 | = | 7 | ALA4423300 | 7.00 | nM | Rattus norvegicus | |||
14. | Eplerenone | 1 | pIC50 | = | 7.4 | ALA4423300 | 7.40 | nM | Rattus norvegicus | |||
15. | ALA2181928 | 8 | IC50 | = | 3.2 | nM | ALA4028187 | 8.49 | nM | Rattus norvegicus | ||
16. | ALA4086138 | 6aj | IC50 | < | 500 | nM | ALA4008039 | nM | Rattus norvegicus | |||
17. | ALA4064627 | 6ai | IC50 | < | 500 | nM | ALA4008039 | nM | Rattus norvegicus | |||
18. | ALA4082663 | 6ah | IC50 | < | 500 | nM | ALA4008039 | nM | Rattus norvegicus | |||
19. | ALA4060780 | 6ag | IC50 | < | 500 | nM | ALA4008039 | nM | Rattus norvegicus | |||
20. | ALA2181930 | 10, SM-368229 | IC50 | = | 21 | nM | ALA4008038 | 7.68 | nM | Rattus norvegicus |