# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | TH287 | TH287 | IC50 | = | 0.9 | nM | ALA3796259 | 9.05 | nM | Homo sapiens | ||
2. | TH 588 | TH588 | IC50 | = | 7 | nM | ALA3796259 | 8.15 | nM | Homo sapiens | ||
3. | SCH 51344 | 3; SCH51344 | IC50 | = | 410 | nM | ALA3796329 | 6.39 | nM | Homo sapiens | ||
4. | (S)-Crizotinib | 62 | IC50 | = | 330 | nM | ALA3796329 | 6.48 | nM | Homo sapiens | ||
5. | ALA3794167 | 5 | IC50 | = | 0.5 | nM | ALA3796259 | 9.30 | nM | Homo sapiens | ||
6. | ALA3792684 | 6 | IC50 | = | 0.5 | nM | ALA3796259 | 9.30 | nM | Homo sapiens | ||
7. | ALA3794132 | 7 | IC50 | = | 9 | nM | ALA3796259 | 8.05 | nM | Homo sapiens | ||
8. | ALA3780535 | 20 | IC50 | = | 850 | nM | ALA3782419 | 6.07 | nM | Homo sapiens | ||
9. | ALA3780032 | 5; IACS-4759 | Activity | 0 | ALA3783612 | Active | Homo sapiens | |||||
10. | TH 588 | TH588 | INH | 0 | ALA3783609 | Active | % | Homo sapiens | ||||
11. | TH287 | TH287 | INH | 0 | ALA3783609 | Active | % | Homo sapiens | ||||
12. | ALA3780032 | 5; IACS-4759 | INH | 0 | ALA3783609 | Active | % | Homo sapiens | ||||
13. | ALA3781661 | 4; IACS-4619 | INH | 0 | ALA3783609 | Active | % | Homo sapiens | ||||
14. | TH 588 | TH588 | INH | 0 | ALA3783608 | Not Active | % | Homo sapiens | ||||
15. | TH287 | TH287 | INH | 0 | ALA3783608 | Not Active | % | Homo sapiens | ||||
16. | ALA3780032 | 5; IACS-4759 | INH | 0 | ALA3782418 | Active | % | Homo sapiens | ||||
17. | ALA3781661 | 4; IACS-4619 | INH | 0 | ALA3782418 | Active | % | Homo sapiens | ||||
18. | ALA3781493 | 6 | IC50 | = | 112 | nM | ALA3782136 | 6.95 | nM | Homo sapiens | ||
19. | ALA3780652 | 7 | IC50 | = | 302 | nM | ALA3782136 | 6.52 | nM | Homo sapiens | ||
20. | ALA3781296 | 8 | IC50 | = | 22 | nM | ALA3782136 | 7.66 | nM | Homo sapiens |