# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Ageladine A, TFA | ageladine A, 1 | IC50 | = | 0.47 | ug ml-1 | ALA2154854 | ug.mL-1 | Homo sapiens | |||
2. | ALA2153738 | 19 | Ki | > | 200 | uM | ALA2155981 | nM | Homo sapiens | |||
3. | ALA2153739 | 20 | Ki | = | 28 | nM | ALA2155981 | 7.55 | nM | Homo sapiens | ||
4. | ALA3640116 | BDBM100336 | % Ctrl | 109 | % | ALA4887733 | Not Active | % | Homo sapiens | |||
5. | BI 605906 | BI605906 | % Ctrl | 90 | % | ALA4887213 | Not Active | % | Homo sapiens | |||
6. | ALA3337895 | 26f | IC50 | 39 | nM | ALA4883168 | Not Active | nM | Homo sapiens | |||
7. | ALA3337894 | 26c | IC50 | 6.9 | pM | ALA4883157 | Active | nM | Homo sapiens | |||
8. | ALA4588900 | EUB0001182 | % Inhibition of Control Values | 280.8 | % | ALA4882577 | % | Homo sapiens | ||||
9. | ALA1939880 | 19 | IC50 | > | 26 | uM | ALA4882422 | Not Active | nM | Homo sapiens | ||
10. | 4-[[[5-(2-ethoxycarbonyl-1H-indol-5-yl)-1-methylpyrazole-3-carbonyl]amino]methyl]benzoic acid | 15 | IC50 | 1 | nM | ALA4882411 | Active | nM | Homo sapiens | |||
11. | ALA3235416 | 5, BDM43079 | IC50 | > | 100 | uM | ALA3243752 | nM | Homo sapiens | |||
12. | ALA3417764 | 20a | INH | > | 90 | % | ALA3419059 | % | Homo sapiens | |||
13. | ALA3417763 | 19p | INH | > | 90 | % | ALA3419059 | % | Homo sapiens | |||
14. | ALA3417751 | 19d | INH | > | 90 | % | ALA3419059 | % | Homo sapiens | |||
15. | ALA3417745 | 16 | INH | > | 90 | % | ALA3419059 | % | Homo sapiens | |||
16. | ALA3417742 | 13 | INH | > | 90 | % | ALA3419059 | % | Homo sapiens | |||
17. | ALA409502 | 3a | IC50 | = | 32 | uM | ALA3399891 | 4.50 | nM | Homo sapiens | ||
18. | ALA410649 | 3g | IC50 | = | 55.88 | uM | ALA3399891 | 4.25 | nM | Homo sapiens | ||
19. | ALA263909 | 3j | IC50 | = | 25 | uM | ALA3399891 | 4.60 | nM | Homo sapiens | ||
20. | ALA260125 | 3b | IC50 | = | 0.158 | uM | ALA3399891 | 6.80 | nM | Homo sapiens |