# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Marimastat (BB-2516) | 2c (BB-2516) | pIC50 | = | 5 | ALA3761998 | 5.00 | nM | Homo sapiens | |||
2. | ALA424130 | 1f | IC50 | = | 1789 | nM | ALA5119020 | 5.75 | nM | Homo sapiens | ||
3. | ALA475540 | C | Activity | 0 | ALA940657 | Active | Homo sapiens | |||||
4. | ALA500351 | W | Activity | 0 | ALA940657 | Not Active | Homo sapiens | |||||
5. | 2-[(4-Chlorophenyl)methylthio]-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one | K | Activity | 0 | ALA940657 | Not Active | Homo sapiens | |||||
6. | ALA497985 | 51 | IC50 | > | 5000 | nM | ALA1005438 | nM | Homo sapiens | |||
7. | ALA325163 | 12d | Ki | > | 2000 | nM | ALA1005438 | nM | Homo sapiens | |||
8. | IK-862 | IK682 | Ki | = | 3997 | nM | ALA1005438 | 5.40 | nM | Homo sapiens | ||
9. | ALA207305 | 12z | Ki | > | 7088 | nM | ALA1005438 | nM | Homo sapiens | |||
10. | ALA495502 | 36 | Ki | = | 1700 | nM | ALA1005438 | 5.77 | nM | Homo sapiens | ||
11. | ALA253275 | 32 | Ki | > | 10000 | nM | ALA1005438 | nM | Homo sapiens | |||
12. | ALA402393 | 49 | Ki | > | 7088 | nM | ALA1005438 | nM | Homo sapiens | |||
13. | ALA402393 | 49 | Ki | > | 7088 | nM | ALA934166 | nM | Homo sapiens | |||
14. | ALA271235 | 21m | Ki | > | 7100 | nM | ALA930634 | nM | Homo sapiens | |||
15. | ALA447787 | 19 | Ki | > | 7088 | nM | ALA946136 | nM | Homo sapiens | |||
16. | ALA403186 | 17 | Ki | > | 7088 | nM | ALA946136 | nM | Homo sapiens | |||
17. | ALA402436 | 15 | Ki | > | 7088 | nM | ALA946136 | nM | Homo sapiens | |||
18. | ALA603656 | 29b | Ki | > | 25 | uM | ALA1069314 | nM | Homo sapiens | |||
19. | ALA1956115 | 1a | Ki | > | 10 | uM | ALA1960131 | nM | Homo sapiens | |||
20. | ALA234034 | 18 | IC50 | > | 7000 | nM | ALA897392 | nM | Homo sapiens |