# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Marimastat (BB-2516) | 2c (BB-2516) | pIC50 | = | 5 | ALA3761999 | 5.00 | nM | Homo sapiens | |||
2. | ALA424130 | 1f | IC50 | = | 1839 | nM | ALA5119021 | 5.74 | nM | Homo sapiens | ||
3. | ALA4585243 | EUB0000728 | IC50 | = | 940 | nM | ALA5213667 | 6.03 | nM | Homo sapiens | ||
4. | ALA1939846 | 1c | IC50 | = | 39 | nM | ALA1942113 | 7.41 | nM | Homo sapiens | ||
5. | ALA1939845 | 1b | IC50 | = | 2200 | nM | ALA1942113 | 5.66 | nM | Homo sapiens | ||
6. | ALA1939844 | 1a | IC50 | = | 1100 | nM | ALA1942113 | 5.96 | nM | Homo sapiens | ||
7. | ALA475540 | C | Activity | 0 | ALA940658 | Active | Homo sapiens | |||||
8. | ALA500351 | W | Activity | 0 | ALA940658 | Not Active | Homo sapiens | |||||
9. | 2-[(4-Chlorophenyl)methylthio]-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one | K | Activity | 0 | ALA940658 | Not Active | Homo sapiens | |||||
10. | ALA468900 | P01 | Activity | 0 | ALA1005428 | Not Active | Homo sapiens | |||||
11. | ALA325163 | 12d | Ki | > | 2000 | nM | ALA1005436 | nM | Homo sapiens | |||
12. | IK-862 | IK682 | Ki | = | 1599 | nM | ALA1005436 | 5.80 | nM | Homo sapiens | ||
13. | ALA207305 | 12z | Ki | > | 5554 | nM | ALA1005436 | nM | Homo sapiens | |||
14. | ALA253275 | 32 | Ki | > | 10000 | nM | ALA1005436 | nM | Homo sapiens | |||
15. | ALA253275 | 32 | Ki | > | 10000 | nM | ALA946137 | nM | Homo sapiens | |||
16. | ALA447787 | 19 | Ki | > | 5554 | nM | ALA946137 | nM | Homo sapiens | |||
17. | ALA403186 | 17 | Ki | > | 5554 | nM | ALA946137 | nM | Homo sapiens | |||
18. | ALA402436 | 15 | Ki | > | 5454 | nM | ALA946137 | nM | Homo sapiens | |||
19. | ALA603656 | 29b | Ki | > | 25 | uM | ALA1069315 | nM | Homo sapiens | |||
20. | ARP 101 | (R)-5a | IC50 | = | 51 | nM | ALA1042359 | 7.29 | nM | Homo sapiens |