# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5279102 | 21; BAY-805 | IC50 | = | 8.6 | uM | ALA5251195 | 5.07 | nM | Homo sapiens | ||
2. | ALA5279102 | 21; BAY-805 | INH | = | 58 | % | ALA5251194 | % | Homo sapiens | |||
3. | ALA5288241 | B2 | INH | < | 50 | % | ALA5238276 | % | Homo sapiens | |||
4. | BI 2536 | 1 | % of control | = | 86 | % | ALA5213529 | % | Homo sapiens | |||
5. | PF 3644022 | PF-3644022 | IC50 | = | 5 | nM | ALA5210310 | 8.30 | nM | Homo sapiens | ||
6. | PF 3644022 | PF-3644022 | IC50 | = | 159 | nM | ALA5209900 | 6.80 | nM | Homo sapiens | ||
7. | ALA5201686 | 10f | Activity | > | 75 | % | ALA5158122 | % | Homo sapiens | |||
8. | ALA5185001 | 24j | INH | < | 40 | % | ALA5115516 | % | Homo sapiens | |||
9. | ALA4564126 | 18 | INH | <= | 16 | % | ALA4427654 | % | Homo sapiens | |||
10. | ALA4564126 | 18 | IC50 | >= | 5 | uM | ALA4427710 | nM | Homo sapiens | |||
11. | ALA4445335 | Roxyl-ZV-5J | INH | = | 1 | % | ALA4408091 | % | Homo sapiens | |||
12. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405438 | % | Homo sapiens | |||
13. | ALA4559936 | (+/-)-6 | Activity | = | 42 | % | ALA4391427 | % | Homo sapiens | |||
14. | ALA4564973 | 50 | INH | = | 100 | % | ALA4389801 | % | Homo sapiens | |||
15. | ALA4555459 | 43 | INH | = | 100 | % | ALA4389324 | % | Homo sapiens | |||
16. | ALA4545456 | 24 | INH | = | 13.5 | % | ALA4387336 | % | Homo sapiens | |||
17. | Abemaciclib | ABEMACICLIB | INH | = | 5 | % | ALA4387336 | % | Homo sapiens | |||
18. | ALA4473365 | 7c | Activity | = | 100 | % | ALA4382605 | % | Homo sapiens | |||
19. | Dasatinib | 2, BMS-354825 | Activity | > | 75 | % | ALA4807898 | % | Homo sapiens | |||
20. | ALA4855726 | B3 | Activity | > | 75 | % | ALA4807898 | % | Homo sapiens |