# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4846335 | 19b | INH | > | 70 | % | ALA4841130 | % | Rattus norvegicus | |||
2. | Alogliptin | 10, alogliptin, SYR-322 | INH | = | 45 | % | ALA4841130 | % | Rattus norvegicus | |||
3. | ALA4845890 | 19h | INH | > | 70 | % | ALA4841129 | % | Rattus norvegicus | |||
4. | ALA4851477 | 19e | INH | > | 70 | % | ALA4841129 | % | Rattus norvegicus | |||
5. | ALA4846335 | 19b | INH | > | 70 | % | ALA4841129 | % | Rattus norvegicus | |||
6. | ALA4845890 | 19h | INH | = | 90 | % | ALA4841128 | % | Rattus norvegicus | |||
7. | ALA4851477 | 19e | INH | = | 90 | % | ALA4841128 | % | Rattus norvegicus | |||
8. | ALA4846335 | 19b | INH | = | 90 | % | ALA4841128 | % | Rattus norvegicus | |||
9. | ALA4090635 | 6d | IC50 | = | 4170 | nM | ALA4021428 | 5.38 | nM | Rattus norvegicus | ||
10. | ALA4078112 | 6c | IC50 | = | 1230 | nM | ALA4021428 | 5.91 | nM | Rattus norvegicus | ||
11. | ALA4086264 | 6b | IC50 | = | 319 | nM | ALA4021428 | 6.50 | nM | Rattus norvegicus | ||
12. | ALA4067185 | 6a | IC50 | = | 155 | nM | ALA4021428 | 6.81 | nM | Rattus norvegicus | ||
13. | sitagliptin | Sitagliptin | IC50 | = | 33 | nM | ALA4021428 | 7.48 | nM | Rattus norvegicus | ||
14. | Enalaprilat | 3 | IC50 | 0 | ALA4021428 | Not Determined | Rattus norvegicus | |||||
15. | rac-Sitagliptin | BDBM126822 | IC50 | = | 26.01 | nM | ALA3705997 | 7.58 | 256873 | nM | Rattus norvegicus | |
16. | ALA3665969 | BDBM126821 | IC50 | = | 80.1 | nM | ALA3705997 | 7.10 | 256872 | nM | Rattus norvegicus | |
17. | ALA3665968 | BDBM126820 | IC50 | = | 2.61 | nM | ALA3705997 | 8.58 | 256871 | nM | Rattus norvegicus | |
18. | ALA3665967 | BDBM126819 | IC50 | = | 23.22 | nM | ALA3705997 | 7.63 | 256870 | nM | Rattus norvegicus | |
19. | ALA3665966 | BDBM126818 | IC50 | = | 11.48 | nM | ALA3705997 | 7.94 | 256869 | nM | Rattus norvegicus | |
20. | ALA3665965 | BDBM126817 | IC50 | = | 25.85 | nM | ALA3705997 | 7.59 | 256868 | nM | Rattus norvegicus |