# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3086657 | ENT | t1/2 | = | 5 | min | ALA3090292 | hr | Rattus norvegicus | |||
2. | rac-Sitagliptin | BDBM126822 | IC50 | = | 26.01 | nM | ALA3705997 | 7.58 | 256873 | nM | Rattus norvegicus | |
3. | ALA3665969 | BDBM126821 | IC50 | = | 80.1 | nM | ALA3705997 | 7.10 | 256872 | nM | Rattus norvegicus | |
4. | ALA3665968 | BDBM126820 | IC50 | = | 2.61 | nM | ALA3705997 | 8.58 | 256871 | nM | Rattus norvegicus | |
5. | ALA3665967 | BDBM126819 | IC50 | = | 23.22 | nM | ALA3705997 | 7.63 | 256870 | nM | Rattus norvegicus | |
6. | ALA3665966 | BDBM126818 | IC50 | = | 11.48 | nM | ALA3705997 | 7.94 | 256869 | nM | Rattus norvegicus | |
7. | ALA3665965 | BDBM126817 | IC50 | = | 25.85 | nM | ALA3705997 | 7.59 | 256868 | nM | Rattus norvegicus | |
8. | ALA3665964 | BDBM126816 | IC50 | = | 11.2 | nM | ALA3705997 | 7.95 | 256867 | nM | Rattus norvegicus | |
9. | ALA3665963 | BDBM126815 | IC50 | = | 17.7 | nM | ALA3705997 | 7.75 | 256866 | nM | Rattus norvegicus | |
10. | ALA3665962 | BDBM126814 | IC50 | = | 22.83 | nM | ALA3705997 | 7.64 | 256865 | nM | Rattus norvegicus | |
11. | ALA4846335 | 19b | INH | > | 70 | % | ALA4841130 | % | Rattus norvegicus | |||
12. | Alogliptin | 10, alogliptin, SYR-322 | INH | = | 45 | % | ALA4841130 | % | Rattus norvegicus | |||
13. | ALA4845890 | 19h | INH | > | 70 | % | ALA4841129 | % | Rattus norvegicus | |||
14. | ALA4851477 | 19e | INH | > | 70 | % | ALA4841129 | % | Rattus norvegicus | |||
15. | ALA4846335 | 19b | INH | > | 70 | % | ALA4841129 | % | Rattus norvegicus | |||
16. | ALA4845890 | 19h | INH | = | 90 | % | ALA4841128 | % | Rattus norvegicus | |||
17. | ALA4851477 | 19e | INH | = | 90 | % | ALA4841128 | % | Rattus norvegicus | |||
18. | ALA4846335 | 19b | INH | = | 90 | % | ALA4841128 | % | Rattus norvegicus | |||
19. | ALA4090635 | 6d | IC50 | = | 4170 | nM | ALA4021428 | 5.38 | nM | Rattus norvegicus | ||
20. | ALA4078112 | 6c | IC50 | = | 1230 | nM | ALA4021428 | 5.91 | nM | Rattus norvegicus |