# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278465 | 33 | IC50 | > | 2 | uM | ALA5252868 | nM | Homo sapiens | |||
2. | ALA5288565 | 29 | IC50 | > | 2 | uM | ALA5252868 | nM | Homo sapiens | |||
3. | ALA5270581 | 18 | IC50 | > | 2 | uM | ALA5252868 | nM | Homo sapiens | |||
4. | ALA1951346 | 36 | IC50 | = | 62 | nM | ALA5244639 | 7.21 | nM | Homo sapiens | ||
5. | ALA5286659 | 44 | IC50 | = | 18 | nM | ALA5244639 | 7.75 | nM | Homo sapiens | ||
6. | ALA5286659 | 44 | IC50 | = | 781 | uM | ALA5244632 | nM | Homo sapiens | |||
7. | ALA3613623 | 26 | IC50 | > | 1000 | nM | ALA5244632 | nM | Homo sapiens | |||
8. | ALA3613600 | 3 | IC50 | = | 8.9 | nM | ALA5244632 | 8.05 | nM | Homo sapiens | ||
9. | ALA3613598 | 1 | IC50 | < | 1 | nM | ALA5244632 | nM | Homo sapiens | |||
10. | LX7101 | 28, LX7101 | IC50 | = | 340 | nM | ALA5244632 | 6.47 | nM | Homo sapiens | ||
11. | ALA3797874 | 3 | IC50 | > | 1000 | nM | ALA5244632 | nM | Homo sapiens | |||
12. | ALA3799326 | 2 | IC50 | > | 1000 | nM | ALA5244632 | nM | Homo sapiens | |||
13. | ALA5267815 | 12a | INH | 0 | ALA5244015 | Not Active | % | Homo sapiens | ||||
14. | netarsudil | NETARSUDIL | Ki | = | 2 | nM | ALA5242770 | 8.70 | nM | Homo sapiens | ||
15. | AR-13324 M1 metabolite | 13 | Ki | = | 0.2 | nmol/L | ALA5242767 | 9.70 | nM | Homo sapiens | ||
16. | netarsudil | NETARSUDIL | Ki | = | 1 | nmol/L | ALA5242767 | 9.00 | nM | Homo sapiens | ||
17. | ripasudil | ripasudil | IC50 | = | 0.019 | uM | ALA5242765 | 7.72 | nM | Homo sapiens | ||
18. | ALA269538 | 1 | IC50 | > | 40 | uM | ALA5235539 | nM | Homo sapiens | |||
19. | ALA4594302 | 17 | IC50 | = | 105 | nM | ALA5228484 | 6.98 | nM | Homo sapiens | ||
20. | ALA5278924 | 14 | IC50 | = | 2100 | nM | ALA5228482 | 5.68 | nM | Homo sapiens |