# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | artepillin C | 5 | IC50 | = | 350000 | nM | ALA5241295 | nM | Homo sapiens | |||
2. | ALA5286645 | 19 | Ki | = | 9400 | nM | ALA5241291 | 5.03 | nM | Homo sapiens | ||
3. | ALA4301261 | 17; ND-336 | Ki | = | 120 | nM | ALA5241291 | 6.92 | nM | Homo sapiens | ||
4. | ALA5281328 | 16 | Ki | = | 40 | nM | ALA5241291 | 7.40 | nM | Homo sapiens | ||
5. | ALA1834423 | 13, M4 | Ki | = | 260 | nM | ALA5241291 | 6.58 | nM | Homo sapiens | ||
6. | ALA1834422 | 3, ND-322 | Ki | = | 100 | nM | ALA5241291 | 7.00 | nM | Homo sapiens | ||
7. | ALA2380403 | 29f | Ki | = | 5 | nM | ALA5241291 | 8.30 | nM | Homo sapiens | ||
8. | ALA2380401 | 29c | Ki | = | 62 | nM | ALA5241291 | 7.21 | nM | Homo sapiens | ||
9. | ALA4859268 | 53 | IC50 | > | 200000 | nM | ALA5237966 | nM | Homo sapiens | |||
10. | ALA5287253 | 64 | INH | = | 22.3 | % | ALA5234320 | % | Homo sapiens | |||
11. | ALA5277375 | Compound 31; 22 | IC50 | = | 56.33 | uM | ALA5232270 | 4.25 | nM | Homo sapiens | ||
12. | Rebimastat | 3, BMS-275291 | IC50 | = | 40 | nM | ALA5232270 | 7.40 | nM | Homo sapiens | ||
13. | Batimastat | 2d (BB-94) | IC50 | = | 2.9 | nM | ALA5232270 | 8.54 | nM | Homo sapiens | ||
14. | ALA2431028 | 21 | IC50 | = | 19500 | nM | ALA5229263 | 4.71 | nM | Homo sapiens | ||
15. | ALA5276957 | 3 | IC50 | = | 234000 | nM | ALA5229263 | nM | Homo sapiens | |||
16. | ALA5283335 | 2 | IC50 | = | 50000 | nM | ALA5229263 | 4.30 | nM | Homo sapiens | ||
17. | ALA5267938 | 1 | IC50 | = | 57000 | nM | ALA5229263 | 4.24 | nM | Homo sapiens | ||
18. | ALA5220395 | 20 | INH | 0 | ALA5217301 | NA | % | Homo sapiens | ||||
19. | ALA5219770 | 19 | INH | 0 | ALA5217301 | NA | % | Homo sapiens | ||||
20. | ALA5219237 | 18 | INH | 0 | ALA5217301 | NA | % | Homo sapiens |