# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Neratinib (HKI-272) | 25o (table 3) | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
2. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
3. | AZD8055 | 10, AZD-8055 | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
4. | Dasatinib | 2, BMS-354825 | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
5. | Axitinib | AG-13736 | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
6. | ALA1614701 | AZD-6244 | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
7. | Poziotinib (HM781-36B) | POZIOTINIB | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
8. | Gilteritinib | GILTERITINIB | Kd apparent | = | 451 | nM | ALA3991882 | 6.35 | Active | nM | Homo sapiens | |
9. | ALA3688339 | BDBM166063 | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
10. | Erlotinib | Tarceva | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
11. | Vandetanib | 22 | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
12. | AMG-208 | 4 | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
13. | Bafetinib (INNO-406) | 9b | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
14. | BI 2536 | 1 | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
15. | Tucatinib (Irbinitinib, ONT-380) | TUCATINIB | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
16. | ALA3545328 | XL-019 | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
17. | Tivantinib (ARQ 197) | TIVANTINIB | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
18. | Fostamatinib (R788) | FOSTAMATINIB | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
19. | SU 14813 | SU-14813 | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens | ||
20. | JANEX-1 | JANEX-1 | Kd apparent | > | 30000 | nM | ALA3991882 | Inactive | nM | Homo sapiens |