# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Bazedoxifene | 7 ; TSE-424 | INH | 0 | ALA3776543 | Active | % | Homo sapiens | ||||
2. | Raloxifene | 44 | INH | 0 | ALA3776543 | Active | % | Homo sapiens | ||||
3. | clomiphene | 1 | INH | 0 | ALA3776543 | Active | % | Homo sapiens | ||||
4. | Tamoxifen | Tamoxifen | INH | 0 | ALA3776543 | Active | % | Homo sapiens | ||||
5. | L-Centchroman | 1-l (l-Centchroman) | INH | 0 | ALA3776543 | Active | % | Homo sapiens | ||||
6. | Toremifene | Toremifene | INH | 0 | ALA3776553 | Active | % | Homo sapiens | ||||
7. | ALA5281526 | 25; TASIN-32 | IC50 | = | 0.049 | uM | ALA5226845 | 7.31 | nM | Homo sapiens | ||
8. | ALA5284923 | 24; TASIN-18 | IC50 | < | 1 | uM | ALA5226845 | nM | Homo sapiens | |||
9. | ALA5270628 | 23; TASIN-38 | IC50 | = | 188 | nM | ALA5226845 | 6.73 | nM | Homo sapiens | ||
10. | ALA4544901 | 47; ww2-83 | IC50 | = | 97.3 | nM | ALA5226845 | 7.01 | nM | Homo sapiens | ||
11. | ALA5285995 | 21; TASIN-35 | IC50 | = | 2.95 | nM | ALA5226845 | 8.53 | nM | Homo sapiens | ||
12. | ALA4454956 | 103; ww1-224 | IC50 | = | 9.36 | nM | ALA5226845 | 8.03 | nM | Homo sapiens | ||
13. | ALA5285729 | 19; TASIN-21 | IC50 | = | 303 | nM | ALA5226845 | 6.52 | nM | Homo sapiens | ||
14. | ALA4091520 | (+/-)-3b | INH | 0 | ALA4035568 | Active | % | Homo sapiens | ||||
15. | ALA3828326 | 18e | INH | 0 | ALA4035568 | Active | % | Homo sapiens | ||||
16. | ALA3827403 | 18c | INH | 0 | ALA4035568 | Active | % | Homo sapiens | ||||
17. | ALA4091520 | (+/-)-3b | INH | 0 | ALA4035569 | Not Active | % | Homo sapiens | ||||
18. | ALA3828326 | 18e | INH | 0 | ALA4035569 | Not Active | % | Homo sapiens | ||||
19. | ALA3827403 | 18c | INH | 0 | ALA4035569 | Not Active | % | Homo sapiens | ||||
20. | ALA2311153 | [11C]SA4503 | Ki | = | 1.7 | nM | ALA2186107 | 8.77 | nM | Homo sapiens |