# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Remibrutinib (LOU064) | 25; LOU064 | Activity | 0 | ALA4358601 | Not Active | Homo sapiens | |||||
2. | ALA3480577 | DDD01251909 | Mean fold stimulation | 0.35 | ALA4883487 | Homo sapiens | ||||||
3. | ALA3401466 | AmBF3-MJ9 | Ki | = | 0.5 | nM | ALA3407092 | 9.30 | nM | Homo sapiens | ||
4. | ALA3401466 | AmBF3-MJ9 | IC50 | = | 0.6 | nM | ALA3407092 | 9.22 | nM | Homo sapiens | ||
5. | ALA3401467 | 18F-AmBF3-MJ9 | Activity | = | 5.48 | % | ALA3407094 | % | Homo sapiens | |||
6. | ALA3401467 | 18F-AmBF3-MJ9 | Activity | = | 5.84 | % | ALA3407095 | % | Homo sapiens | |||
7. | ALA3401467 | 18F-AmBF3-MJ9 | Activity | = | 5.32 | % | ALA3407096 | % | Homo sapiens | |||
8. | ALA3401467 | 18F-AmBF3-MJ9 | Activity | = | 2.37 | % | ALA3407097 | % | Homo sapiens | |||
9. | ALA3401467 | 18F-AmBF3-MJ9 | Activity | = | 1.54 | % | ALA3407098 | % | Homo sapiens | |||
10. | ALA3947545 | [125I]-Tyr(4)-BBN | Activity | 0 | ALA3880110 | Active | Homo sapiens | |||||
11. | ALA3961428 | [125I]-[DTyr(6), betaAlan(11), Phe(13), Nle(14)]-BBN(6-14) | Activity | 0 | ALA3880110 | Active | Homo sapiens | |||||
12. | ALA3967904 | Table 16, R1C2 | IC50 | = | 2.2 | nM | ALA3880106 | 8.66 | nM | Homo sapiens | ||
13. | ALA3963000 | Table 14, R7C2 | IC50 | = | 366 | nM | ALA3880106 | 6.44 | nM | Homo sapiens | ||
14. | ALA3984233 | L300 | IC50 | = | 2.5 | nM | ALA3880106 | 8.60 | nM | Homo sapiens | ||
15. | ALA3944194 | Table 13, R19C2, Table 14, R2C2 | IC50 | = | 450 | nM | ALA3880106 | 6.35 | nM | Homo sapiens | ||
16. | ALA3928975 | L228 | IC50 | = | 5.5 | nM | ALA3880106 | 8.26 | nM | Homo sapiens | ||
17. | ALA3890803 | L227 | IC50 | = | 28 | nM | ALA3880106 | 7.55 | nM | Homo sapiens | ||
18. | ALA3975022 | L226 | IC50 | = | 5.5 | nM | ALA3880106 | 8.26 | nM | Homo sapiens | ||
19. | ALA3932925 | L225 | IC50 | = | 240 | nM | ALA3880106 | 6.62 | nM | Homo sapiens | ||
20. | ALA3935631 | L224 | IC50 | = | 52 | nM | ALA3880106 | 7.28 | nM | Homo sapiens |