# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Lanceolatin B | 10a | IC50 | > | 20 | uM | ALA4675245 | nM | Homo sapiens | |||
2. | ALA577397 | 4 | IC50 | > | 20 | uM | ALA4675245 | nM | Homo sapiens | |||
3. | ALA3542381 | M20 | Drug metabolism | 0 | ALA3532129 | metabolite_detected | Homo sapiens | |||||
4. | ALA3542336 | [14C]-SCH 530348 | Drug metabolism | 0 | ALA3529575 | metabolite_detected | Homo sapiens | |||||
5. | Panobinostat (LBH589) | 5, LBH-589 | Stability | = | 56 | % | ALA3537637 | % | Homo sapiens | |||
6. | ALA3526395 | M1 | Drug metabolism | = | 3.2 | % | ALA3537638 | % | Homo sapiens | |||
7. | ALA3526396 | M2 | Drug metabolism | = | 2.6 | % | ALA3537638 | % | Homo sapiens | |||
8. | ALA3526818 | [14C]-Fingolimod, FTY720 | Drug metabolism | 0 | ALA3533010 | metabolite_not_detected | Homo sapiens | |||||
9. | ALA3527525 | M4 | Drug metabolism | = | 38 | % | ALA3537638 | % | Homo sapiens | |||
10. | ALA3527526 | M5 | Drug metabolism | = | 0.1 | % | ALA3537638 | % | Homo sapiens | |||
11. | ALA42 | clozapine | Drug metabolism | = | 4.08 | nmol/min | ALA3538130 | nmol/min | Homo sapiens | |||
12. | ALA42 | clozapine | Drug metabolism | = | 5.71 | nmol/min | ALA3541788 | nmol/min | Homo sapiens | |||
13. | ALA42 | clozapine | Drug metabolism | = | 0.025 | nmol/min | ALA3539709 | nmol/min | Homo sapiens | |||
14. | ALA42 | clozapine | Drug metabolism | = | 0.065 | nmol/min | ALA3539720 | nmol/min | Homo sapiens | |||
15. | ALA42 | clozapine | Drug metabolism | = | 0.41 | nmol/min | ALA3536203 | nmol/min | Homo sapiens | |||
16. | oxymetazoline | Oxymetazoline | Drug metabolism | 0 | ALA3535091 | metabolite_not_detected | Homo sapiens | |||||
17. | oxymetazoline | Oxymetazoline | Drug metabolism | 0 | ALA3530226 | metabolite_not_detected | Homo sapiens | |||||
18. | MCC950 | SID144210780 | Drug metabolism | = | 1.3 | % | ALA3864044 | % | Homo sapiens | |||
19. | ALA120183 | 8 | IC50 | = | 8 | uM | ALA660380 | 5.10 | nM | Homo sapiens | ||
20. | Sulfaphenazole | 29 | IC50 | = | 60 | uM | ALA660380 | 4.22 | nM | Homo sapiens |