| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2130955 | SID85201013 | INH | < | 25 | % | ALA5115435 | % | Homo sapiens | |||
| 2. | ALA2130955 | SID85201013 | IC50 | = | 50 | uM | ALA5115434 | 4.30 | nM | Homo sapiens | ||
| 3. |  8-(benzotriazol-1-ylamino)octanoic acid | 7 | Ratio IC50 | = | 1.6 | ALA4406428 | Homo sapiens | |||||
| 4. |  ALA4442292 | 6 | Ratio IC50 | = | 2.9 | ALA4406428 | Homo sapiens | |||||
| 5. | 8-(benzotriazol-1-ylamino)octanoic acid | 7 | IC50 | = | 179 | uM | ALA4406434 | nM | Homo sapiens | |||
| 6. | ALA4442292 | 6 | IC50 | = | 455 | uM | ALA4406434 | nM | Homo sapiens | |||
| 7. | 8-(benzotriazol-1-ylamino)octanoic acid | 7 | IC50 | = | 282 | uM | ALA4406427 | nM | Homo sapiens | |||
| 8. | ALA4442292 | 6 | IC50 | = | 1330 | uM | ALA4406427 | nM | Homo sapiens | |||
| 9. |  ALA4435658 | 9 | INH | 0 | ALA4406421 | Active | % | Homo sapiens | ||||
| 10. |  ALA4590991 | 8 | INH | 0 | ALA4406421 | Active | % | Homo sapiens | ||||
| 11. | 8-(benzotriazol-1-ylamino)octanoic acid | 7 | INH | 0 | ALA4406421 | Active | % | Homo sapiens | ||||
| 12. | ALA4442292 | 6 | INH | 0 | ALA4406421 | Active | % | Homo sapiens | ||||
| 13. |  ALA3542381 | M20 | Drug metabolism | 0 | ALA3532134 | metabolite_detected | Homo sapiens | |||||
| 14. |  ALA3542336 | [14C]-SCH 530348 | Drug metabolism | 0 | ALA3529775 | metabolite_detected | Homo sapiens | |||||
| 15. |  Panobinostat (LBH589) | 5, LBH-589 | Stability | = | 59 | % | ALA3538476 | % | Homo sapiens | |||
| 16. |  ALA3526395 | M1 | Drug metabolism | = | 2 | % | ALA3538477 | % | Homo sapiens | |||
| 17. |  ALA3526396 | M2 | Drug metabolism | = | 1.5 | % | ALA3538477 | % | Homo sapiens | |||
| 18. |  ALA3526818 | [14C]-Fingolimod, FTY720 | Drug metabolism | 0 | ALA3533015 | metabolite_not_detected | Homo sapiens | |||||
| 19. |  ALA3527525 | M4 | Drug metabolism | = | 37 | % | ALA3538477 | % | Homo sapiens | |||
| 20. |  ALA3526952 | MI | Drug metabolism | = | 0.48 | pmol/min | ALA3528397 | pmol/min | Homo sapiens |
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