# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Ginsenoside Rh2 | 20(S)-Rh2 | Drug metabolism | 0 | ALA3536228 | metabolite_not_detected | Homo sapiens | |||||
2. | ALA3526952 | MI | Vmax(app) | = | 2.57 | pmol/mg.min | ALA3528381 | pmol/mg.min | Homo sapiens | |||
3. | ALA3526952 | MI | Vmax/Km | = | 0.031 | uL/min.mg | ALA3535404 | uL/min.mg | Homo sapiens | |||
4. | ALA3526952 | MI | Km(app) | = | 82.7 | uM | ALA3528381 | nM | Homo sapiens | |||
5. | ALA3527525 | M4 | Drug metabolism | = | 37 | % | ALA3538477 | % | Homo sapiens | |||
6. | ALA3526952 | MI | Drug metabolism | = | 0.48 | pmol/min | ALA3528397 | pmol/min | Homo sapiens | |||
7. | ALA3542381 | M20 | Drug metabolism | 0 | ALA3532134 | metabolite_detected | Homo sapiens | |||||
8. | ALA3542336 | [14C]-SCH 530348 | Drug metabolism | 0 | ALA3529775 | metabolite_detected | Homo sapiens | |||||
9. | Panobinostat (LBH589) | 5, LBH-589 | Stability | = | 59 | % | ALA3538476 | % | Homo sapiens | |||
10. | ALA3526395 | M1 | Drug metabolism | = | 2 | % | ALA3538477 | % | Homo sapiens | |||
11. | ALA3526396 | M2 | Drug metabolism | = | 1.5 | % | ALA3538477 | % | Homo sapiens | |||
12. | ALA3526818 | [14C]-Fingolimod, FTY720 | Drug metabolism | 0 | ALA3533015 | metabolite_not_detected | Homo sapiens | |||||
13. | 8-(benzotriazol-1-ylamino)octanoic acid | 7 | Ratio IC50 | = | 1.6 | ALA4406428 | Homo sapiens | |||||
14. | ALA4442292 | 6 | Ratio IC50 | = | 2.9 | ALA4406428 | Homo sapiens | |||||
15. | 8-(benzotriazol-1-ylamino)octanoic acid | 7 | IC50 | = | 179 | uM | ALA4406434 | nM | Homo sapiens | |||
16. | ALA4442292 | 6 | IC50 | = | 455 | uM | ALA4406434 | nM | Homo sapiens | |||
17. | 8-(benzotriazol-1-ylamino)octanoic acid | 7 | IC50 | = | 282 | uM | ALA4406427 | nM | Homo sapiens | |||
18. | ALA4442292 | 6 | IC50 | = | 1330 | uM | ALA4406427 | nM | Homo sapiens | |||
19. | ALA4435658 | 9 | INH | 0 | ALA4406421 | Active | % | Homo sapiens | ||||
20. | ALA4590991 | 8 | INH | 0 | ALA4406421 | Active | % | Homo sapiens |