# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4202767 | 56 | Activity | <= | 25 | % | ALA4187167 | % | Homo sapiens | |||
2. | [³H]valsartan | valsartan | pIC50 | 0 | ALA4311876 | Not Determined | Homo sapiens | |||||
3. | ALA4435800 | 35; TD-0212 | pIC50 | = | 7.1 | ALA4311876 | 7.10 | nM | Homo sapiens | |||
4. | Omapatrilat | 1a, BMS-186716 | pIC50 | 0 | ALA4311876 | Not Determined | Homo sapiens | |||||
5. | ALA3235416 | 5, BDM43079 | IC50 | > | 100 | uM | ALA3243747 | nM | Homo sapiens | |||
6. | ALA3222111 | 27b | pIC50 | < | 4.5 | ALA3223376 | nM | Homo sapiens | ||||
7. | ALA3221965 | 27a | pIC50 | < | 4.5 | ALA3223376 | nM | Homo sapiens | ||||
8. | ALA3221964 | 22b | pIC50 | < | 4.5 | ALA3223376 | nM | Homo sapiens | ||||
9. | ALA3221963 | 22a | pIC50 | < | 4.5 | ALA3223376 | nM | Homo sapiens | ||||
10. | Selective PI3Kδ Inhibitor 1 (compound 7n) | 7n | IC50 | > | 0.3 | uM | ALA4001595 | nM | Homo sapiens | |||
11. | ALA3640116 | BDBM100336 | % Ctrl | 82 | % | ALA4887718 | Not Active | % | Homo sapiens | |||
12. | BI 605906 | BI605906 | % Ctrl | 82 | % | ALA4887199 | Not Active | % | Homo sapiens | |||
13. | PQCA | 4i | % inhibition | 45 | % | ALA4882998 | Not Active | % | Homo sapiens | |||
14. | PPTN | 2 | % inhibition | 12 | % | ALA4882998 | Not Active | % | Homo sapiens | |||
15. | ALA4588900 | EUB0001182 | % Inhibition of Control Values | 14.3 | % | ALA4882551 | % | Homo sapiens | ||||
16. | BI-1935 | EUB0000542 | % Ctrl | 84 | % | ALA4882513 | Not Active | % | Homo sapiens | |||
17. | ALA4633785 | 35 | IC50 | = | 431 | uM | ALA4617715 | nM | Homo sapiens | |||
18. | ALA4520267 | 9a | IC50(app) | > | 100 | uM | ALA4480334 | nM | Homo sapiens | |||
19. | ALA4590201 | 8e | IC50(app) | > | 100 | uM | ALA4480334 | nM | Homo sapiens | |||
20. | Z-FA-FMK | 9c | IC50(app) | > | 100 | uM | ALA4480334 | nM | Homo sapiens |