# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Vorinostat (SAHA, MK0683) | SAHA | IC50 | = | 30 | nM | ALA3778485 | 7.52 | nM | Homo sapiens | ||
2. | Panobinostat (LBH589) | 5, LBH-589 | IC50 | = | 2 | nM | ALA3778485 | 8.70 | nM | Homo sapiens | ||
3. | Rocilinostat (ACY-1215) | RICOLINOSTAT | IC50 | = | 135 | nM | ALA3778485 | 6.87 | nM | Homo sapiens | ||
4. | SKLB-23bb | 23bb | IC50 | = | 439 | nM | ALA3778485 | 6.36 | nM | Homo sapiens | ||
5. | (S)-ARN2508 | (+)-10r | Activity | = | -4.3 | % | ALA3777467 | % | Homo sapiens | |||
6. | ALA3769491 | 14a | IC50 | = | 13.7 | uM | ALA3771935 | 4.86 | nM | Homo sapiens | ||
7. | ALA3769629 | 25a | IC50 | > | 30 | uM | ALA3771935 | nM | Homo sapiens | |||
8. | Entinostat (MS-275) | MS-275 | IC50 | = | 0.79 | uM | ALA3771938 | 6.10 | nM | Homo sapiens | ||
9. | ALA1173445 | 4a | IC50 | = | 1.36 | uM | ALA3771942 | 5.87 | nM | Homo sapiens | ||
10. | PCI-34051 | PCI34051 | IC50 | > | 30 | uM | ALA3772307 | nM | Homo sapiens | |||
11. | Vorinostat (SAHA, MK0683) | SAHA | IC50 | = | 0.001 | uM | ALA3772311 | 8.85 | nM | Homo sapiens | ||
12. | ALA3771206 | SD-L-256 | IC50 | = | 0.47 | uM | ALA3772311 | 6.33 | nM | Homo sapiens | ||
13. | HDAC3-IN-T247 | 78, T247 | IC50 | = | 3.94 | uM | ALA3772315 | 5.41 | nM | Homo sapiens | ||
14. | ALA99 | TSA | IC50 | = | 0.02 | uM | ALA3772319 | 7.70 | nM | Homo sapiens | ||
15. | ALA3771288 | 13 | IC50 | = | 65.08 | nM | ALA3774116 | 7.19 | nM | Homo sapiens | ||
16. | ALA3770555 | 12 | IC50 | = | 26.76 | nM | ALA3774116 | 7.57 | nM | Homo sapiens | ||
17. | ALA3770504 | 11 | IC50 | = | 20.79 | nM | ALA3774116 | 7.68 | nM | Homo sapiens | ||
18. | ALA3771366 | 10 | IC50 | = | 113.45 | nM | ALA3774116 | 6.95 | nM | Homo sapiens | ||
19. | ALA3770531 | 9 | IC50 | = | 151.45 | nM | ALA3774116 | 6.82 | nM | Homo sapiens | ||
20. | ALA3769815 | 8 | IC50 | > | 10 | uM | ALA3774116 | nM | Homo sapiens |