# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5273533 | 37 | IC50 | > | 1000 | nM | ALA5244419 | nM | Homo sapiens | |||
2. | ALA5281283 | 18 | IC50 | > | 1000 | nM | ALA5244419 | nM | Homo sapiens | |||
3. | 2,4,3′,5′-tetramethoxystilbene | 7a | INH | 0 | ALA5240278 | Active | % | Homo sapiens | ||||
4. | ALA5280088 | 77 | INH | 0 | ALA5240277 | Active | % | Homo sapiens | ||||
5. | Defactinib | DEFACTINIB | IC50 | = | 3.9 | nM | ALA5238039 | 8.41 | nM | Homo sapiens | ||
6. | PROTAC FAK degrader 1 | Example 102 | IC50 | = | 6.5 | nM | ALA5238039 | 8.19 | nM | Homo sapiens | ||
7. | PROTAC FAK degrader 1 | Example 102 | Emax | = | 99 | % | ALA5238038 | % | Homo sapiens | |||
8. | PROTAC FAK degrader 1 | Example 102 | EC50 | = | 3 | nM | ALA5238037 | 8.52 | nM | Homo sapiens | ||
9. | ALA4518706 | EUB0000702 | % of control | = | 4.9 | % | ALA5213323 | % | Homo sapiens | |||
10. | Lorlatinib | 8k, PF-06463922 | Ki | = | 17 | nM | ALA5213168 | 7.77 | nM | Homo sapiens | ||
11. | XMD8-92 | 18 | IC50 | = | 39 | uM | ALA5213125 | 4.41 | nM | Homo sapiens | ||
12. | MPS1-IN-1 | Mps1-IN-1 | IC50 | = | 440 | nM | ALA5212779 | 6.36 | nM | Homo sapiens | ||
13. | ALA4540759 | EUB0000545 | % of control | = | 17 | % | ALA5214560 | % | Homo sapiens | |||
14. | Defactinib | DEFACTINIB | IC50 | = | 0.2 | nM | ALA5210428 | 9.70 | nM | Homo sapiens | ||
15. | ALA4518706 | EUB0000702 | IC50 | = | 721 | nM | ALA5210416 | 6.14 | nM | Homo sapiens | ||
16. | Defactinib | DEFACTINIB | IC50 | = | 3 | nM | ALA5210174 | 8.52 | nM | Homo sapiens | ||
17. | ALA5184634 | 7m | INH | 0 | ALA5160595 | Dde | % | Homo sapiens | ||||
18. | ALA5184634 | 7m | INH | 0 | ALA5160594 | Dde | % | Homo sapiens | ||||
19. | ALA5206391 | 2l | INH | = | 0 | % | ALA5159002 | % | Homo sapiens | |||
20. | ALA5170735 | 2k | INH | = | 0 | % | ALA5159002 | % | Homo sapiens |