# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | NMS-E973 | 18, NMS-E973 | IC50 | > | 10 | nM | ALA2444007 | nM | Homo sapiens | |||
2. | ALA2443138 | 30 | IC50 | > | 10 | nM | ALA2444007 | nM | Homo sapiens | |||
3. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2444007 | nM | Homo sapiens | |||
4. | ALA2443026 | 38 | IC50 | > | 10 | nM | ALA2444007 | nM | Homo sapiens | |||
5. | NVP-TAE 226 | 1a, TAE226 | IC50 | = | 5.5 | nM | ALA2432167 | 8.26 | nM | Homo sapiens | ||
6. | PF-573228 | PF-228 | IC50 | = | 4 | nM/L | ALA2432167 | 8.40 | nM | Homo sapiens | ||
7. | PF-00562271 | PF-562,271 | IC50 | = | 1.5 | nmol/L | ALA2432166 | 8.82 | nM | Homo sapiens | ||
8. | PND-1186 hydrochloride | PND-1186 | IC50 | = | 1.5 | nM | ALA2432164 | 8.82 | nM | Homo sapiens | ||
9. | ALA2425654 | 3 | INH | < | 50 | % | ALA2429478 | % | Homo sapiens | |||
10. | ALA2425652 | 4 | INH | < | 50 | % | ALA2429478 | % | Homo sapiens | |||
11. | ALA2425649 | 8 | INH | < | 50 | % | ALA2429478 | % | Homo sapiens | |||
12. | ALA2425645 | 11 | INH | < | 50 | % | ALA2429478 | % | Homo sapiens | |||
13. | ALA2425644 | 13 | INH | = | 85 | % | ALA2429478 | % | Homo sapiens | |||
14. | PF-562271 | PF-562271 | IC50 | = | 1.5 | nM | ALA2427453 | 8.82 | nM | Homo sapiens | ||
15. | N-(5-chloropyridin-2-yl)acetamide | 1 | Kd | = | 719 | uM | ALA2427451 | 3.14 | nM | Homo sapiens | ||
16. | 4-(Pyridin-3-yl)pyrimidin-2-amine | 1 | Kd | = | 159 | uM | ALA2427451 | 3.80 | nM | Homo sapiens | ||
17. | 5-(5-Bromo-3-pyridyl)-1H-tetrazole | 3 | Kd | = | 95 | uM | ALA2427451 | 4.02 | nM | Homo sapiens | ||
18. | 5-(4-Pyridyl)-1,3-oxazole | 15 | Kd | = | 1350 | uM | ALA2427451 | 2.87 | nM | Homo sapiens | ||
19. | ALA2315560 | 1 | Kd | = | 43 | uM | ALA2427451 | 4.37 | nM | Homo sapiens | ||
20. | ALA1599242 | SID858265 | Kd | = | 93 | uM | ALA2427451 | 4.03 | nM | Homo sapiens |