# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | β-Estradiol | Table II | IC50 | = | 8.7 | nM | ALA2330135 | 8.06 | nM | Homo sapiens | ||
2. | ALA2326072 | 14, J1 | IC50 | = | 19.1 | nM | ALA2330135 | 7.72 | nM | Homo sapiens | ||
3. | ALA2326073 | 16, J2 | IC50 | = | 120.7 | nM | ALA2330135 | 6.92 | nM | Homo sapiens | ||
4. | ALA2326074 | 11, J3 | IC50 | = | 331.1 | nM | ALA2330135 | 6.48 | nM | Homo sapiens | ||
5. | ALA2326075 | 10, J4 | IC50 | = | 436.4 | nM | ALA2330135 | 6.36 | nM | Homo sapiens | ||
6. | ALA2326076 | 12, J5 | IC50 | = | 185 | nM | ALA2330135 | 6.73 | nM | Homo sapiens | ||
7. | ALA2326071 | 15, J6 | IC50 | = | 565.9 | nM | ALA2330135 | 6.25 | nM | Homo sapiens | ||
8. | ALA2326070 | 17, J7 | IC50 | = | 111.9 | nM | ALA2330135 | 6.95 | nM | Homo sapiens | ||
9. | ALA2326069 | 13, J8 | IC50 | = | 150.6 | nM | ALA2330135 | 6.82 | nM | Homo sapiens | ||
10. | ALA2326068 | 18, J9 | IC50 | = | 41.2 | nM | ALA2330135 | 7.38 | nM | Homo sapiens | ||
11. | ALA2326072 | 14, J1 | RBA | = | 45.7 | % | ALA2330133 | % | Homo sapiens | |||
12. | ALA2326073 | 16, J2 | RBA | = | 7.2 | % | ALA2330133 | % | Homo sapiens | |||
13. | ALA2326074 | 11, J3 | RBA | = | 2.6 | % | ALA2330133 | % | Homo sapiens | |||
14. | ALA2326075 | 10, J4 | RBA | = | 2 | % | ALA2330133 | % | Homo sapiens | |||
15. | ALA2326076 | 12, J5 | RBA | = | 4.7 | % | ALA2330133 | % | Homo sapiens | |||
16. | ALA2326071 | 15, J6 | RBA | = | 1.5 | % | ALA2330133 | % | Homo sapiens | |||
17. | ALA2326070 | 17, J7 | RBA | = | 7.8 | % | ALA2330133 | % | Homo sapiens | |||
18. | ALA2326069 | 13, J8 | RBA | = | 5.8 | % | ALA2330133 | % | Homo sapiens | |||
19. | ALA2326068 | 18, J9 | RBA | = | 21.1 | % | ALA2330133 | % | Homo sapiens | |||
20. | ALA4776913 | 1 | Activity | < | 10 | % | ALA4715116 | % | Homo sapiens |