# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA353846 | adiphenine | pIC50 | = | 4.77 | ALA2169535 | 4.77 | nM | Rattus norvegicus | |||
2. | Chlorprothixene | 32 | pIC50 | = | 8.97 | ALA2169535 | 8.97 | nM | Rattus norvegicus | |||
3. | ALA596 | 1 (fentanyl) | pIC50 | = | 4.7 | ALA2169535 | 4.70 | nM | Rattus norvegicus | |||
4. | mepyramine | Mepyramine | pIC50 | = | 8.24 | ALA2169535 | 8.24 | nM | Rattus norvegicus | |||
5. | Orphenadrine | orphenadrine | pIC50 | = | 6.79 | ALA2169535 | 6.79 | nM | Rattus norvegicus | |||
6. | procyclidine | 147 | pIC50 | = | 5.17 | ALA2169535 | 5.17 | nM | Rattus norvegicus | |||
7. | promazine | promazine | pIC50 | = | 5.9 | ALA2169535 | 5.90 | nM | Rattus norvegicus | |||
8. | Phentolamine | Phentolamine | pIC50 | = | 4.9 | ALA2169535 | 4.90 | nM | Rattus norvegicus | |||
9. | ALA2103769 | 16 | pIC50 | = | 4.95 | ALA2169535 | 4.95 | nM | Rattus norvegicus | |||
10. | ALA1277935 | 48, stereoisomer2 | pKi | = | 8.06 | ALA1287099 | 8.06 | nM | Rattus norvegicus | |||
11. | ALA1277770 | 51 | pKi | = | 8.33 | ALA1287099 | 8.33 | nM | Rattus norvegicus | |||
12. | ALA1277678 | 54 | pKi | = | 7.91 | ALA1287099 | 7.91 | nM | Rattus norvegicus | |||
13. | ALA1276947 | 64 | pKi | = | 8.27 | ALA1287099 | 8.27 | nM | Rattus norvegicus | |||
14. | ALA1276948 | 65 | pKi | = | 8.25 | ALA1287099 | 8.25 | nM | Rattus norvegicus | |||
15. | ALA1277126 | 69 | pKi | = | 7.7 | ALA1287099 | 7.70 | nM | Rattus norvegicus | |||
16. | ALA1277312 | 73 | pKi | = | 7.85 | ALA1287099 | 7.85 | nM | Rattus norvegicus | |||
17. | ALA1935574 | 66, VUF11489 | Ki | = | 3600 | nM | ALA1936682 | 5.44 | nM | Rattus norvegicus | ||
18. | ALA274768 | 11 | Emax | = | 0 | ALA697087 | Rattus norvegicus | |||||
19. | ALA274768 | 11 | Emax | = | 0 | ALA697087 | Rattus norvegicus | |||||
20. | ALA274768 | 11 | Relative potency | = | 5.72 | ALA697088 | Rattus norvegicus |