# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4166126 | QC-308 | IC50 | = | 0.46 | uM | ALA4433389 | 6.34 | nM | Homo sapiens | ||
2. | ALA1187207 | 5 | IC50 | > | 100 | uM | ALA4433389 | nM | Homo sapiens | |||
3. | ALA482686 | I-90 | IC50 | = | 2.2 | uM | ALA4433389 | 5.66 | nM | Homo sapiens | ||
4. | OB 24 hydrochloride | 7c | IC50 | > | 100 | uM | ALA4433389 | nM | Homo sapiens | |||
5. | ALA4756381 | 7 | Activity | 0 | ALA4672537 | Active | Homo sapiens | |||||
6. | ARS-1620 | ARS-1620, (S)-Atropisomer | IC50 | = | 7.64 | uM | ALA4721807 | 5.12 | nM | Homo sapiens | ||
7. | ARS-1620 | ARS-1620, (S)-Atropisomer | Ratio | = | -0.3 | ALA4721797 | Homo sapiens | |||||
8. | JNJ-38877605 | SID137276033 | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens | ||
9. | RGB-286638 | RGB-286638 | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens | ||
10. | Apatinib | SID124955476 | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens | ||
11. | Temsirolimus (CCI-779, NSC 683864) | Temsirolimus | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens | ||
12. | Sunitinib | 12b | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens | ||
13. | Barasertib (AZD1152-HQPA) | 34 | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens | ||
14. | AZD5363 | 64, AZD5363 | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens | ||
15. | SCIO 469 hydrochloride | SCIO-469 | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens | ||
16. | AZD5438 | 6 | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens | ||
17. | Y-33075 | 23, Y-39983 | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens | ||
18. | Linifanib (ABT-869) | 17p, ABT-869 | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens | ||
19. | Dinaciclib (SCH727965) | DINACICLIB | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens | ||
20. | Imatinib (STI571) | 1 | Kd apparent | > | 30000 | nM | ALA3991731 | Inactive | nM | Homo sapiens |