# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4533775 | 22 | Ki | = | 460 | nM | ALA4478055 | 6.34 | nM | Homo sapiens | ||
2. | ALA4581302 | 21 | Ki | > | 10000 | nM | ALA4478055 | nM | Homo sapiens | |||
3. | ALA4581256 | 20 | Ki | = | 220 | nM | ALA4478055 | 6.66 | nM | Homo sapiens | ||
4. | ALA4576579 | 19 | Ki | = | 550 | nM | ALA4478055 | 6.26 | nM | Homo sapiens | ||
5. | ALA3787713 | 18 | Ki | = | 220 | nM | ALA4478055 | 6.66 | nM | Homo sapiens | ||
6. | ALA3787712 | 17 | Ki | = | 140 | nM | ALA4478055 | 6.85 | nM | Homo sapiens | ||
7. | ALA3787766 | 16 | Ki | = | 280 | nM | ALA4478055 | 6.55 | nM | Homo sapiens | ||
8. | ALA4549208 | (2S,7S)-10 | Ki | = | 400 | nM | ALA4478055 | 6.40 | nM | Homo sapiens | ||
9. | ALA4522438 | (2R,7R)-10 | Ki | = | 710 | nM | ALA4478055 | 6.15 | nM | Homo sapiens | ||
10. | ALA4475071 | (S,S)-1 | Ki | = | 2100 | nM | ALA4478055 | 5.68 | nM | Homo sapiens | ||
11. | ALA4456247 | (R,R)-1 | Ki | = | 1500 | nM | ALA4478055 | 5.82 | nM | Homo sapiens | ||
12. | (S)-VU0637120 | VU0673120 | INH | 0 | ALA4738237 | Not Active | % | Homo sapiens | ||||
13. | ALA4277590 | 39 | pEC50 | = | 8.5 | ALA4265260 | 8.50 | nM | Homo sapiens | |||
14. | ALA4277590 | 39 | pKi | = | 9.2 | ALA4265256 | 9.20 | nM | Homo sapiens | |||
15. | ALA4277590 | 39 | EC50 | = | 3.2 | nM | ALA4265260 | 8.49 | nM | Homo sapiens | ||
16. | ALA4277590 | 39 | Ki | = | 0.63 | nM | ALA4265256 | 9.20 | nM | Homo sapiens | ||
17. | ALA4294418 | 38 | pEC50 | = | 6.4 | ALA4265260 | 6.40 | nM | Homo sapiens | |||
18. | ALA4294418 | 38 | pKi | = | 6.1 | ALA4265256 | 6.10 | nM | Homo sapiens | |||
19. | ALA4294418 | 38 | EC50 | = | 400 | nM | ALA4265260 | 6.40 | nM | Homo sapiens | ||
20. | ALA4294418 | 38 | Ki | = | 790 | nM | ALA4265256 | 6.10 | nM | Homo sapiens |