# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | LDC1267 | 7; LDC1267 | % of control | < | 10 | % | ALA5212926 | % | Homo sapiens | |||
2. | BMS-777607 | 10, BMS-777607 | IC50 | = | 1.8 | nM | ALA5210326 | 8.74 | nM | Homo sapiens | ||
3. | BMS-777607 | 10, BMS-777607 | IC50 | = | 150 | nM | ALA5209912 | 6.82 | nM | Homo sapiens | ||
4. | ALA4445335 | Roxyl-ZV-5J | INH | = | 54 | % | ALA4408119 | % | Homo sapiens | |||
5. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405549 | % | Homo sapiens | |||
6. | ALA4559936 | (+/-)-6 | Activity | = | 89 | % | ALA4391455 | % | Homo sapiens | |||
7. | ALA4564973 | 50 | INH | = | 100 | % | ALA4389829 | % | Homo sapiens | |||
8. | ALA4555459 | 43 | INH | = | 100 | % | ALA4389352 | % | Homo sapiens | |||
9. | ALA4545456 | 24 | INH | = | 7 | % | ALA4387349 | % | Homo sapiens | |||
10. | Abemaciclib | ABEMACICLIB | INH | = | 10.5 | % | ALA4387349 | % | Homo sapiens | |||
11. | ALA4473365 | 7c | Activity | = | 100 | % | ALA4382633 | % | Homo sapiens | |||
12. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379420 | nM | Homo sapiens | |||
13. | CDK9-IN-7 | 21e | INH | = | 72 | % | ALA4377847 | % | Homo sapiens | |||
14. | ALA4584949 | 23a | INH | = | 50 | % | ALA4376564 | % | Homo sapiens | |||
15. | ALA4584949 | 23a | IC50 | = | 346 | nM | ALA4376518 | 6.46 | nM | Homo sapiens | ||
16. | Dasatinib | 2, BMS-354825 | Activity | > | 75 | % | ALA4807987 | % | Homo sapiens | |||
17. | ALA4855726 | B3 | Activity | > | 75 | % | ALA4807987 | % | Homo sapiens | |||
18. | ALA4867844 | C7 | Activity | > | 75 | % | ALA4807987 | % | Homo sapiens | |||
19. | ALA2348350 | 15u | Activity | = | 99 | % | ALA4806642 | % | Homo sapiens | |||
20. | ALA2348350 | 15u | Activity | = | 97 | % | ALA4806642 | % | Homo sapiens |