# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5283294 | 48 | IC50 | = | 4.69 | nM | ALA5237507 | 8.33 | nM | Homo sapiens | ||
2. | Roflumilast | table 2 Roflumilast (17) | IC50 | = | 3 | nM | ALA5236726 | 8.52 | nM | Homo sapiens | ||
3. | ALA511115 | 1 (Ariflo) | IC50 | = | 813 | nM | ALA5236726 | 6.09 | nM | Homo sapiens | ||
4. | 4-[8-(2,1,3-Benzoxadiazol-5-yl)-1,7-naphthyridin-6-yl]benzoic acid | 1 | IC50 | = | 1.23 | nM | ALA5236726 | nM | Homo sapiens | |||
5. | ALA4867572 | 4r | IC50 | = | 1.25 | uM | ALA5216831 | 5.90 | nM | Homo sapiens | ||
6. | BPN14770 | ZATOLMILAST | INH | 0 | ALA4397288 | Not Active | % | Homo sapiens | ||||
7. | [³H]rolipram | 1 | INH | = | 70 | % | ALA4395095 | % | Homo sapiens | |||
8. | ALA4584299 | 3t | INH | = | 20 | % | ALA4395094 | % | Homo sapiens | |||
9. | ALA4468513 | 3b; DRILS-1765 | INH | = | 20 | % | ALA4395094 | % | Homo sapiens | |||
10. | ALA4783529 | 11h | INH | < | 50 | % | ALA4730669 | % | Homo sapiens | |||
11. | Ibudilast | Ibudilast | IC50 | = | 239 | nM | ALA4725707 | 6.62 | nM | Homo sapiens | ||
12. | ALA4784887 | 18-2 | IC50 | = | 3 | nM | ALA4725687 | 8.52 | nM | Homo sapiens | ||
13. | ALA4752341 | 18-3 | IC50 | = | 3 | nM | ALA4725687 | 8.52 | nM | Homo sapiens | ||
14. | ALA4750999 | 18-4 | IC50 | = | 3 | nM | ALA4725687 | 8.52 | nM | Homo sapiens | ||
15. | ALA4787980 | 18-6 | IC50 | = | 3 | nM | ALA4725687 | 8.52 | nM | Homo sapiens | ||
16. | ALA4757093 | 18-5 | IC50 | = | 3 | nM | ALA4725687 | 8.52 | nM | Homo sapiens | ||
17. | ALA4759270 | 18-1 | IC50 | = | 3 | nM | ALA4725687 | 8.52 | nM | Homo sapiens | ||
18. | ALA4762291 | 5 | IC50 | = | 1100 | nM | ALA4709044 | 5.96 | nM | Homo sapiens | ||
19. | CP-671305 | SID144210764 | IC50 | = | 3858 | nM | ALA4709041 | 5.41 | nM | Homo sapiens | ||
20. | [³H]rolipram | 1 | IC50 | = | 1258 | nM | ALA4709041 | 5.90 | nM | Homo sapiens |