# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Trabodenoson | TRABODENOSON | K | = | 0.97 | nM | ALA5242773 | nM | Homo sapiens | |||
2. | ALA5280210 | 31 | INH | = | 61 | % | ALA5236909 | % | Homo sapiens | |||
3. | ALA4788488 | 16; MRS7334, PDSP 44294 | Ki | > | 10000 | nM | ALA5233323 | nM | Homo sapiens | |||
4. | ALA3612932 | 12 | Ki | > | 10000 | nM | ALA5233323 | nM | Homo sapiens | |||
5. | ALA11048 | 44 | Ki | = | 3 | uM | ALA5223713 | 5.52 | nM | Homo sapiens | ||
6. | 8(p-Sulfophenyl)theophylline | 6a (SPT) | Ki | = | 4.5 | uM | ALA5223713 | 5.35 | nM | Homo sapiens | ||
7. | KW 3902 | 2 (KW-3902) | Ki | = | 1.3 | nM | ALA5223711 | 8.89 | nM | Homo sapiens | ||
8. | [³H]XAC | 4 | Kd | = | 0.17 | nM | ALA5223707 | 9.77 | nM | Homo sapiens | ||
9. | 1,3-Diethyl-8-phenylxanthine | 1 | IC50 | = | 1 | uM | ALA5223705 | 6.00 | nM | Homo sapiens | ||
10. | 1,3-Dimethyl-8-phenylxanthine | 10a | IC50 | = | 0.5 | uM | ALA5223705 | 6.30 | nM | Homo sapiens | ||
11. | ALA158077 | 12 | Ki | = | 6.5 | nM | ALA5223693 | 8.19 | nM | Homo sapiens | ||
12. | ALA11002 | 73 | Ki | = | 6.5 | nM | ALA5223693 | 8.19 | nM | Homo sapiens | ||
13. | ALA298474 | 8 | Ki | = | 0.95 | nM | ALA5223693 | 9.02 | nM | Homo sapiens | ||
14. | Caffeine | caffeine | pKi | = | 4.3 | ALA5223688 | 4.30 | nM | Homo sapiens | |||
15. | Caffeine | caffeine | IC50 | = | 10.7 | uM | ALA5223688 | 4.97 | nM | Homo sapiens | ||
16. | Theobromine | theobromine | IC50 | = | 105 | uM | ALA5223688 | nM | Homo sapiens | |||
17. | Theobromine | theobromine | Ki | = | 105 | uM | ALA5223683 | nM | Homo sapiens | |||
18. | OF-1 | 8 | % of inhibition | = | 82 | % | ALA5214231 | % | Homo sapiens | |||
19. | BAY-299 | 5b; atropisomer 2 | % of control | = | 48 | % | ALA5214107 | % | Homo sapiens | |||
20. | A 196 | A-196 | Ki | = | 12 | nM | ALA5214590 | 7.92 | nM | Homo sapiens |