# | Name | Compound Key | Action Type | Relation | Activety Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PD184352 (CI-1040) | 1 | Kd | = | 120 | nM | ALA1908590 | 6.92 | nM | Homo sapiens | ||
2. | Barasertib (AZD1152-HQPA) | 34 | Kd | = | 1900 | nM | ALA1908590 | 5.72 | nM | Homo sapiens | ||
3. | Pazopanib | 13 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
4. | GW2580 (DMSO solution) | K00591a, Diaminopyrimidine1 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
5. | Canertinib (CI-1033) | 18 | Kd | = | 1800 | nM | ALA1908590 | 5.75 | nM | Homo sapiens | ||
6. | AT7519 | 33 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
7. | Sorafenib | 5 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
8. | Nilotinib (AMN-107) | 38 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
9. | GSK690693 | 3g, GSK-690693 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
10. | RAF265 (CHIR-265) | CHIR-265/RAF-265 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
11. | AST-487 (NVP-AST487) | AST-487 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
12. | Bosutinib Isomer 1, Free Base | 1 (SKI-606) | Kd | = | 19 | nM | ALA1908590 | 7.72 | nM | Homo sapiens | ||
13. | MLN8054 | MLN-8054 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
14. | GSK461364 | GSK-461364A | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
15. | ALA522892 | 5 | Kd | = | 520 | nM | ALA1908590 | 6.28 | nM | Homo sapiens | ||
16. | SGX-523 | SGX-523 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
17. | Tandutinib (MLN518) | 75 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
18. | GSK1838705A | 40 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
19. | Motesanib | AMG-706 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens | |||
20. | SB-203580 | 9 | Kd | > | 10000 | nM | ALA1908590 | nM | Homo sapiens |