# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5288212 | 7a | INH | 0 | ALA5251456 | Not Active | % | Homo sapiens | ||||
2. | ALA5271471 | 6 | IC50 | > | 16 | uM | ALA5248063 | nM | Homo sapiens | |||
3. | ALA5279683 | 23 | IC50 | > | 30 | uM | ALA5239624 | nM | Homo sapiens | |||
4. | opnurasib | 1a | INH | = | 12 | % | ALA5238528 | % | Homo sapiens | |||
5. | opnurasib | 1a | IC50 | > | 10 | uM | ALA5238526 | nM | Homo sapiens | |||
6. | GX 201 | 14; GX-201 | IC50 | = | 3.2 | nM | ALA5225022 | 8.49 | nM | Homo sapiens | ||
7. | ALA4471012 | 13; GX-585 | IC50 | = | 435 | nM | ALA5225022 | 6.36 | nM | Homo sapiens | ||
8. | ALA5289676 | 29 | IC50 | > | 33000 | nM | ALA5225017 | nM | Homo sapiens | |||
9. | ALA3945969 | BDBM217483 | IC50 | > | 14000 | nM | ALA5225011 | nM | Homo sapiens | |||
10. | Funapide | FUNAPIDE | IC50 | = | 0.084 | uM | ALA5224991 | 7.08 | nM | Homo sapiens | ||
11. | Raxatrigine | VIXOTRIGINE | IC50 | = | 3.2 | uM | ALA5224988 | 5.50 | nM | Homo sapiens | ||
12. | Carbamazepine | carbamazepine | IC50 | = | 46.8 | uM | ALA5224988 | 4.33 | nM | Homo sapiens | ||
13. | ALA5275826 | 13 | IC50 | > | 100 | uM | ALA5224985 | nM | Homo sapiens | |||
14. | mexiletine | Mexiletine | IC50 | = | 15 | uM | ALA5224985 | 4.82 | nM | Homo sapiens | ||
15. | ALA79 | 1 | IC50 | = | 50 | uM | ALA5224985 | 4.30 | nM | Homo sapiens | ||
16. | ALA5178575 | 28; ARUK3001185 | IC50 | > | 30 | uM | ALA5166943 | nM | Homo sapiens | |||
17. | ALA5200705 | 26 | INH | = | 7.7 | % | ALA5164182 | % | Homo sapiens | |||
18. | ALA5190568 | 48 | IC50 | > | 30 | uM | ALA5154400 | nM | Homo sapiens | |||
19. | ALA5198935 | 30-distomer | INH | 0 | ALA5154206 | NA | % | Homo sapiens | ||||
20. | GDC-0077 | INAVOLISIB | INH | < | 20 | % | ALA5153895 | % | Homo sapiens |