# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Tetraethylthiuram disulfide | disulfiram | pIC50 | = | 4.4 | ALA1046622 | 4.40 | nM | Rattus norvegicus | |||
2. | EWP 815 | 10 | pIC50 | = | 4.8 | ALA1046622 | 4.80 | nM | Rattus norvegicus | |||
3. | ALA494494 | 2 | IC50 | = | 0.72 | uM | ALA960209 | 6.14 | nM | Rattus norvegicus | ||
4. | ALA449188 | 1 | IC50 | = | 0.36 | uM | ALA960209 | 6.44 | nM | Rattus norvegicus | ||
5. | N-Methyl-N-propargylbenzylamine | Pargyline | IC50 | = | 5.6 | uM | ALA960209 | 5.25 | nM | Rattus norvegicus | ||
6. | ALA455595 | psi(epsilon)RACK | Activity | = | 3.2 | micromol/min | ALA1019411 | micromol/min | Rattus norvegicus | |||
7. | ALA455595 | psi(epsilon)RACK | Activity | = | 33 | % | ALA1019408 | % | Rattus norvegicus | |||
8. | ALA455595 | psi(epsilon)RACK | Activity | 0 | ALA1019408 | Active | Rattus norvegicus | |||||
9. | ALA294687 | 6 | Inhibition | 0 | % | ALA646618 | % | Rattus norvegicus | ||||
10. | ALA282540 | 1b | AIDH activity | = | 19 | nM min-1 | ALA660110 | nM min-1 | Rattus norvegicus | |||
11. | ALA282540 | 1b | AIDH activity | = | 13.4 | nM min-1 | ALA660109 | nM min-1 | Rattus norvegicus | |||
12. | ALA282540 | 1b | Inhibition | = | 73.7 | % | ALA660113 | % | Rattus norvegicus | |||
13. | ALA282540 | 1b | Inhibition | = | 48.9 | % | ALA660112 | % | Rattus norvegicus | |||
14. | Chlorpropamide | Chloropropamide | AlDH activity | = | 73.8 | nM min-1 | ALA660111 | nM min-1 | Rattus norvegicus | |||
15. | Chlorpropamide | Chloropropamide | AIDH activity | = | 28.3 | nM min-1 | ALA660109 | nM min-1 | Rattus norvegicus | |||
16. | Chlorpropamide | Chloropropamide | Inhibition | = | 0 | % | ALA660113 | % | Rattus norvegicus | |||
17. | Chlorpropamide | Chloropropamide | Inhibition | = | 0 | % | ALA660112 | % | Rattus norvegicus | |||
18. | ALA299785 | 1c | Inhibition | 0 | % | ALA646617 | % | Rattus norvegicus |