# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3771118 | 4a; PF-06761281 | pIC50 | = | 5 | ALA3773094 | 5.00 | nM | Homo sapiens | |||
2. | ALA3771118 | 4a; PF-06761281 | IC50 | = | 14.1 | uM | ALA3773094 | 4.85 | nM | Homo sapiens | ||
3. | PF-06761281 | 1a; PF-06649298 | IC50 | > | 100 | uM | ALA3773094 | nM | Homo sapiens | |||
4. | ALA1686 | alpha-ketoglutarate | EC50 | = | 54 | uM | ALA5209627 | 4.27 | Substrate | nM | Homo sapiens | |
5. | Succinic acid | Succinic acid | EC50 | = | 107 | uM | ALA5209627 | Substrate | nM | Homo sapiens |