# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Lapatinib | GW-572016 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
2. | AZD8931 (Sapitinib) | 2, AZD8931 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
3. | P276-00 | P-276-00 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
4. | AZD2014 | 21, AZD2014 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
5. | ALA1822792 | MK-2461 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
6. | Bafetinib (INNO-406) | 9b | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
7. | Foretinib (GSK1363089) | EXEL-2880/GSK-1363089 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
8. | Ponatinib (AP24534) | 20g, AP24534 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
9. | EMD 1214063 | 22 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
10. | LGX 818 | ENCORAFENIB | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
11. | LY2801653 | MERESTINIB | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
12. | TG02 (Double bond E) | 26h, SB1317/TG02 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
13. | AT7519 | 33 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
14. | CP-724714 | 4 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
15. | Amuvatinib (MP-470) | AMUVATINIB | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
16. | SAR407899 | 14C | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
17. | AZD1208 | 28 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
18. | RGB-286638 | RGB-286638 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
19. | Fostamatinib (R788) | FOSTAMATINIB | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens | ||
20. | CEP-32496 | 40, CEP-32496 | Kd apparent | > | 30000 | nM | ALA3991924 | Inactive | nM | Homo sapiens |