# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4585117 | 1 | Drug metabolism | = | 30 | % | ALA4477629 | % | Homo sapiens | |||
2. | ALA4585117 | 1 | t1/2 | = | 49.5 | min | ALA4477630 | hr | Homo sapiens | |||
3. | ALA4585117 | 1 | Drug metabolism | = | 55.8 | pmol/min | ALA4477631 | pmol/min | Homo sapiens | |||
4. | ALA1422005 | SID26729800 | t1/2 | = | 99 | min | ALA4419284 | hr | Homo sapiens | |||
5. | loperamide | Loperamide | Ki | = | 1.5 | uM | ALA4711507 | 5.82 | nM | Homo sapiens | ||
6. | ALA4776624 | B5 | INH | 0 | ALA4711504 | Dose-dependent effect | % | Homo sapiens | ||||
7. | ALA4776624 | B5 | IC50 | = | 4.45 | uM | ALA4711504 | 5.35 | nM | Homo sapiens | ||
8. | ALA4776624 | B5 | Ki | = | 0.068 | uM | ALA4711503 | 7.17 | nM | Homo sapiens | ||
9. | loperamide | Loperamide | IC50 | = | 6.8 | uM | ALA4711500 | 5.17 | nM | Homo sapiens | ||
10. | ALA4780848 | B10 | IC50 | = | 0.63 | uM | ALA4711500 | 6.20 | nM | Homo sapiens | ||
11. | ALA4748399 | B6 | IC50 | = | 0.38 | uM | ALA4711500 | 6.42 | nM | Homo sapiens | ||
12. | ALA4748929 | B8 | IC50 | = | 0.81 | uM | ALA4711500 | 6.09 | nM | Homo sapiens | ||
13. | ALA4776624 | B5 | IC50 | = | 0.052 | uM | ALA4711500 | 7.28 | nM | Homo sapiens | ||
14. | ALA4740149 | B4 | IC50 | = | 0.61 | uM | ALA4711500 | 6.21 | nM | Homo sapiens | ||
15. | ALA4745825 | B3 | IC50 | = | 2.86 | uM | ALA4711500 | 5.54 | nM | Homo sapiens | ||
16. | ALA4752404 | B2 | IC50 | = | 1.62 | uM | ALA4711500 | 5.79 | nM | Homo sapiens | ||
17. | ALA4756815 | B1 | IC50 | = | 2.91 | uM | ALA4711500 | 5.54 | nM | Homo sapiens | ||
18. | ALA4751728 | A4 | IC50 | = | 1.48 | uM | ALA4711500 | 5.83 | nM | Homo sapiens | ||
19. | ALA4761197 | A1 | IC50 | = | 1.31 | uM | ALA4711500 | 5.88 | nM | Homo sapiens | ||
20. | ALA4747287 | A3 | IC50 | = | 1.09 | uM | ALA4711500 | 5.96 | nM | Homo sapiens |