# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA175257 | Ac-NH-Asp-Tyr(SO3H)-Nle-NH2 | Ki | = | 5 | uM | ALA5246400 | 5.30 | nM | Rattus norvegicus | ||
2. | PTP1B-IN-2 | P6 | Activity | = | 38.1 | % | ALA3826031 | % | Rattus norvegicus | |||
3. | ALA3823340 | P4 | Activity | = | 27.7 | % | ALA3826031 | % | Rattus norvegicus | |||
4. | PTP1B-IN-2 | P6 | Activity | = | 19 | % | ALA3826030 | % | Rattus norvegicus | |||
5. | ALA3823340 | P4 | Activity | = | 26.1 | % | ALA3826030 | % | Rattus norvegicus | |||
6. | PTP1B-IN-2 | P6 | Activity | = | 16 | % | ALA3826029 | % | Rattus norvegicus | |||
7. | ALA3823340 | P4 | Activity | = | 6.9 | % | ALA3826029 | % | Rattus norvegicus | |||
8. | ALA2296205 | 14a | INH | = | 25.3 | % | ALA3074012 | % | Rattus norvegicus | |||
9. | ALA2296206 | 14b | INH | = | 38.5 | % | ALA3074012 | % | Rattus norvegicus | |||
10. | ALA2296207 | 14c | INH | = | 13.5 | % | ALA3074012 | % | Rattus norvegicus | |||
11. | ALA2296208 | 14d | INH | = | 26.6 | % | ALA3074012 | % | Rattus norvegicus | |||
12. | ALA2296209 | 14e | INH | = | 24.2 | % | ALA3074012 | % | Rattus norvegicus | |||
13. | ALA2296210 | 14f | INH | = | 13.3 | % | ALA3074012 | % | Rattus norvegicus | |||
14. | ALA2296211 | 14g | INH | = | 18.8 | % | ALA3074012 | % | Rattus norvegicus | |||
15. | ALA2296212 | 14h | INH | = | 11.8 | % | ALA3074012 | % | Rattus norvegicus | |||
16. | N,N-Dimethylimidodicarbonimidic diamide | Metformine | INH | = | 30.2 | % | ALA3074012 | % | Rattus norvegicus | |||
17. | ALA121 | BRL-49653 | INH | = | 25.2 | % | ALA3074012 | % | Rattus norvegicus | |||
18. | ALA2282786 | ZINC02765569 | INH | = | 18.5 | % | ALA3077716 | % | Rattus norvegicus | |||
19. | ALA121 | BRL-49653 | INH | = | 25.2 | % | ALA3077715 | % | Rattus norvegicus | |||
20. | N,N-Dimethylimidodicarbonimidic diamide | Metformine | INH | = | 30.2 | % | ALA3077714 | % | Rattus norvegicus |