# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5288951 | Cyclo-MG2 | IC50 | = | 3.23 | nM | ALA5241823 | 8.49 | nM | Homo sapiens | ||
2. | ALA5273681 | Cyclo-MG1 | IC50 | = | 2.54 | nM | ALA5241823 | 8.60 | nM | Homo sapiens | ||
3. | PF 05105679 | 8, PF-05105679 | % of effect | = | 35 | % | ALA5214512 | % | Homo sapiens | |||
4. | ALA5177923 | Leu15-gastrin-17 | EC50 | = | 2.4 | nM | ALA5146166 | 8.62 | nM | Homo sapiens | ||
5. | ALA5205878 | xGLP-1 | EC50 | 0 | ALA5146166 | ND | Homo sapiens | |||||
6. | ALA410972 | 1 | EC50 | 0 | ALA5146166 | ND | Homo sapiens | |||||
7. | ALA5182775 | 2d | EC50 | > | 100 | nM | ALA5146166 | nM | Homo sapiens | |||
8. | ALA5182331 | 2c | EC50 | > | 100 | nM | ALA5146166 | nM | Homo sapiens | |||
9. | ALA5182323 | 2b | EC50 | > | 100 | nM | ALA5146166 | nM | Homo sapiens | |||
10. | ALA5181266 | 2a | EC50 | > | 100 | nM | ALA5146166 | nM | Homo sapiens | |||
11. | ALA5185239 | 1b | EC50 | > | 100 | nM | ALA5146166 | nM | Homo sapiens | |||
12. | ALA5182173 | 1a | EC50 | > | 100 | nM | ALA5146166 | nM | Homo sapiens | |||
13. | ALA4440419 | 9; NN9056 | EC50 | > | 100 | nM | ALA5146166 | nM | Homo sapiens | |||
14. | ALA4518377 | Page no 1411, R62C2, cpd 3-(31-Ser) | pEC50 | 0 | ALA4370033 | Not Active | Homo sapiens | |||||
15. | ALA4473611 | Page no 1411, R62C2, cpd 3-(31-Ala) | pEC50 | 0 | ALA4370033 | Not Active | Homo sapiens | |||||
16. | ALA4454469 | Page no 1411, R62C2, cpd 3-(31-Lys) | pEC50 | 0 | ALA4370033 | Not Active | Homo sapiens | |||||
17. | ALA4564249 | Page no 1411, R63C2, cpd 3-(31-Glu) | pEC50 | 0 | ALA4370033 | Not Active | Homo sapiens | |||||
18. | ALA4559510 | Page no 1411, R62C2, cpd 3-(31-Leu) | pEC50 | 0 | ALA4370033 | Active | Homo sapiens | |||||
19. | ALA4590542 | Page no 1412, R23C1, cpd 9-(C-ter-OH) | pEC50 | 0 | ALA4370033 | Not Active | Homo sapiens | |||||
20. | ALA4518377 | Page no 1411, R62C2, cpd 3-(31-Ser) | pIC50 | 0 | ALA4370031 | Not Active | Homo sapiens |