# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GSK065 | 28 | INH | 0 | ALA4051447 | Not Active | % | Homo sapiens | ||||
2. | ALA4064834 | 30; GSK428 | INH | < | 20 | % | ALA4012401 | % | Homo sapiens | |||
3. | PF-04859989 | 7, PF-04859989 | IC50 | = | 30.4 | uM | ALA2329108 | 4.52 | nM | Homo sapiens | ||
4. | ALA2049092 | 19 | IC50 | = | 15.3 | uM | ALA2329108 | 4.82 | nM | Homo sapiens | ||
5. | (3S)-3-amino-1-hydroxy-6-phenoxy-3,4-dihydroquinolin-2-one | 3 | IC50 | = | 2.04 | uM | ALA2329108 | 5.69 | nM | Homo sapiens | ||
6. | ALA2321943 | 4 | IC50 | > | 36 | uM | ALA2329108 | nM | Homo sapiens | |||
7. | PF-04859989 | 7, PF-04859989 | IC50 | = | 22 | uM | ALA2050768 | 4.66 | nM | Homo sapiens | ||
8. | ALA417544 | 4c | Ratio IC50 | = | 7 | ALA1952454 | Homo sapiens | |||||
9. | ALA1950178 | 9f | Ratio IC50 | = | 7 | ALA1952454 | Homo sapiens | |||||
10. | ALA1950173 | 9a | Ratio IC50 | = | 7 | ALA1952454 | Homo sapiens | |||||
11. | ALA1508899 | SID4258075 | IC50 | > | 6000 | uM | ALA1952453 | nM | Homo sapiens | |||
12. | ALA1950317 | 11d | IC50 | > | 1000 | uM | ALA1952453 | nM | Homo sapiens | |||
13. | ALA1950316 | 11c | IC50 | = | 666 | uM | ALA1952453 | nM | Homo sapiens | |||
14. | ALA1950315 | 11b | IC50 | = | 271 | uM | ALA1952453 | nM | Homo sapiens | |||
15. | ALA417544 | 4c | IC50 | = | 293 | uM | ALA1952453 | nM | Homo sapiens | |||
16. | ALA1950179 | 9g | IC50 | = | 34 | uM | ALA1952453 | 4.47 | nM | Homo sapiens | ||
17. | ALA1950178 | 9f | IC50 | = | 20 | uM | ALA1952453 | 4.70 | nM | Homo sapiens | ||
18. | ALA1950177 | 9e | IC50 | = | 43 | uM | ALA1952453 | 4.37 | nM | Homo sapiens | ||
19. | ALA1950176 | 9d | IC50 | = | 33 | uM | ALA1952453 | 4.48 | nM | Homo sapiens | ||
20. | ALA1950173 | 9a | IC50 | = | 20 | uM | ALA1952453 | 4.70 | nM | Homo sapiens |