# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Bexarotene | LGD-1069 | EC50 | 0 | ALA3297478 | Not Determined | Rattus norvegicus | |||||
2. | ALA3289659 | 3 | EC50 | > | 1000 | nM | ALA3297478 | nM | Rattus norvegicus | |||
3. | ALA3289660 | 4 | EC50 | = | 880 | nM | ALA3297478 | 6.06 | nM | Rattus norvegicus | ||
4. | ALA3289657 | 1 | EC50 | = | 440 | nM | ALA3297478 | 6.36 | nM | Rattus norvegicus | ||
5. | ALA3098771 | 9cUAB30, 9-cis-UAB30 | EC50 | = | 400 | nM | ALA3297478 | 6.40 | nM | Rattus norvegicus | ||
6. | ALA3289658 | 2 | EC50 | = | 110 | nM | ALA3297478 | 6.96 | nM | Rattus norvegicus | ||
7. | 9-cis-Retinoic acid | 6 | EC50 | = | 110 | nM | ALA3297478 | 6.96 | nM | Rattus norvegicus | ||
8. | ALA3098773 | (R)-1 | EC50 | = | 19 | nM | ALA3297478 | 7.72 | nM | Rattus norvegicus | ||
9. | 9-cis-Retinoic acid | 6 | EC50 | = | 120 | nM | ALA3100732 | 6.92 | nM | Rattus norvegicus | ||
10. | Bexarotene | LGD-1069 | EC50 | = | 40 | nM | ALA3100732 | 7.40 | nM | Rattus norvegicus | ||
11. | ALA3098771 | 9cUAB30, 9-cis-UAB30 | EC50 | = | 820 | nM | ALA3100732 | 6.09 | nM | Rattus norvegicus | ||
12. | ALA3098772 | (+/-)-1 | EC50 | = | 110 | nM | ALA3100732 | 6.96 | nM | Rattus norvegicus | ||
13. | ALA3098773 | (R)-1 | EC50 | = | 120 | nM | ALA3100732 | 6.92 | nM | Rattus norvegicus | ||
14. | ALA3098858 | (S)-1 | EC50 | = | 120 | nM | ALA3100732 | 6.92 | nM | Rattus norvegicus | ||
15. | ALA337719 | 49 | Synergy | = | 3.1 | fold | ALA878008 | fold | Rattus norvegicus | |||
16. | ALA337719 | 49 | IC50 | = | 2.3 | nM | ALA806515 | 8.64 | nM | Rattus norvegicus | ||
17. | ALA337719 | 49 | Efficacy | = | 79 | % | ALA806513 | % | Rattus norvegicus | |||
18. | ALA337719 | 49 | Efficacy | = | 13 | % | ALA806513 | % | Rattus norvegicus | |||
19. | ALA337719 | 49 | Ki | = | 1 | nM | ALA807181 | 9.00 | nM | Rattus norvegicus | ||
20. | ALA336086 | 25c | Synergy | = | 2.1 | fold | ALA878008 | fold | Rattus norvegicus |