# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | TFB-TBOA | 17b, TFB-TBOA | IC50 | = | 0.2 | uM | ALA5209616 | 6.70 | Inhibitor | nM | Homo sapiens | |
2. | ALA474133 | 1o | IC50 | = | 6.3 | uM | ALA5209616 | 5.20 | Inhibitor | nM | Homo sapiens | |
3. | D-Aspartic acid | 6 (NMDA) | EC50 | = | 398 | uM | ALA5209616 | Substrate | nM | Homo sapiens | ||
4. | L-Aspartic acid | Aspartic acid | EC50 | = | 398 | uM | ALA5209616 | Substrate | nM | Homo sapiens | ||
5. | D-Glutamic acid | gammaCOOH groups in glutamic acid | EC50 | > | 1000 | uM | ALA5209616 | Substrate | nM | Homo sapiens | ||
6. | (S)-(+)-Glutamic acid | Glutamic acid | EC50 | = | 398 | uM | ALA5209616 | Substrate | nM | Homo sapiens | ||
7. | (R)-(+)-Cysteine | Cysteine | EC50 | = | 376 | uM | ALA5209609 | Substrate | nM | Homo sapiens | ||
8. | L-Aspartic acid | Aspartic acid | EC50 | = | 15 | uM | ALA5209609 | 4.82 | Substrate | nM | Homo sapiens | |
9. | (S)-(+)-Glutamic acid | Glutamic acid | EC50 | = | 16 | uM | ALA5209609 | 4.80 | Substrate | nM | Homo sapiens | |
10. | ALA569154 | 10 | INH | 0 | ALA4430907 | Dose-dependent effect | % | Homo sapiens | ||||
11. | ALA4534123 | 4k | pIC50 | < | 3.5 | ALA4430907 | nM | Homo sapiens | ||||
12. | ALA4580984 | 4j | pIC50 | < | 3.5 | ALA4430907 | nM | Homo sapiens | ||||
13. | ALA569154 | 10 | INH | 0 | ALA4430904 | Active | % | Homo sapiens | ||||
14. | ALA569154 | 10 | IC50 | = | 12 | uM | ALA4430907 | 4.92 | nM | Homo sapiens | ||
15. | ALA583892 | 8 | IC50 | > | 300 | uM | ALA4430907 | nM | Homo sapiens | |||
16. | ALA4558690 | 2b | IC50 | > | 300 | uM | ALA4430907 | nM | Homo sapiens | |||
17. | ALA572116 | 3 | IC50 | > | 300 | uM | ALA4430907 | nM | Homo sapiens | |||
18. | ALA4577809 | 2d | IC50 | > | 300 | uM | ALA4430907 | nM | Homo sapiens | |||
19. | ALA4476112 | 2e | IC50 | > | 300 | uM | ALA4430907 | nM | Homo sapiens | |||
20. | ALA4574162 | 3a | IC50 | = | 23 | uM | ALA4430907 | 4.64 | nM | Homo sapiens |