# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3397280 | 286 | INH | = | 100 | % | ALA3399417 | % | Homo sapiens | |||
2. | ALA3397279 | 285 | INH | = | 100 | % | ALA3399416 | % | Homo sapiens | |||
3. | ALA191881 | Leupeptin | Ki | = | 9.2 | uM | ALA3367293 | 5.04 | nM | Homo sapiens | ||
4. | ALA4066494 | 1; A-705253 | INH | = | 84 | % | ALA4041067 | % | Homo sapiens | |||
5. | ALA4287663 | 2b | Ki | = | 1300 | nM | ALA4253884 | 5.89 | nM | Homo sapiens | ||
6. | ALA4279759 | 2a | Ki | 0 | ALA4253884 | Not Active | Homo sapiens | |||||
7. | ALA4292287 | 1b | Ki | = | 7000 | nM | ALA4253884 | 5.16 | nM | Homo sapiens | ||
8. | ALA4292973 | 1a | Ki | 0 | ALA4253884 | Not Active | Homo sapiens | |||||
9. | ALA4287663 | 2b | INH | 0 | ALA4253850 | Not Active | % | Homo sapiens | ||||
10. | ALA4279759 | 2a | INH | 0 | ALA4253850 | Not Active | % | Homo sapiens | ||||
11. | ALA4292287 | 1b | INH | 0 | ALA4253850 | Active | % | Homo sapiens | ||||
12. | ALA4292973 | 1a | INH | 0 | ALA4253850 | Not Active | % | Homo sapiens | ||||
13. | ALA4228126 | 7 | Ki | = | 462 | uM | ALA4221693 | nM | Homo sapiens | |||
14. | ALA4229176 | 15 | Ki | = | 89 | uM | ALA4221696 | 4.05 | nM | Homo sapiens | ||
15. | ALA4229176 | 15 | Ki | = | 89 | uM | ALA4221694 | 4.05 | nM | Homo sapiens | ||
16. | ALA4228921 | 9 | Ki | = | 108 | uM | ALA4221697 | nM | Homo sapiens | |||
17. | ALA4228576 | 8 | Ki | = | 329 | uM | ALA4221694 | nM | Homo sapiens | |||
18. | ALA4228576 | 8 | Ki | = | 329 | uM | ALA4221696 | nM | Homo sapiens | |||
19. | ALA191881 | Leupeptin | Ki | = | 9.2 | uM | ALA3240892 | 5.04 | nM | Homo sapiens | ||
20. | Brensocatib | 30; AZD7986 | IC50 | > | 20 | uM | ALA3859660 | nM | Homo sapiens |