# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Ac-DEVD-CHO,N-Acetyl-Asp-Glu-Val-Asp-al | 2a | IC50 | = | 0.19 | uM | ALA5236703 | 6.72 | nM | Homo sapiens | ||
2. | ALA5280661 | M826 | IC50 | = | 67 | nM | ALA5236703 | 7.17 | nM | Homo sapiens | ||
3. | VRT-043198 | VRT 043198 | Ki | = | 0.8 | nM | ALA5155929 | 9.10 | nM | Homo sapiens | ||
4. | ALA437105 | 2 | IC50 | = | 1.3 | nM | ALA5155929 | 8.89 | nM | Homo sapiens | ||
5. | ALA5173761 | (3R)16ac | Activity | = | 4.45 | % | ALA5155924 | % | Homo sapiens | |||
6. | ALA5206575 | 16ad | Activity | = | 3.9 | % | ALA5155924 | % | Homo sapiens | |||
7. | ALA5172568 | 16ac | Activity | = | 2.91 | % | ALA5155924 | % | Homo sapiens | |||
8. | ALA5175204 | 16ab | Activity | = | 2.06 | % | ALA5155924 | % | Homo sapiens | |||
9. | ALA5185782 | 16aa | Activity | = | 2.47 | % | ALA5155924 | % | Homo sapiens | |||
10. | ALA5204759 | 5ce | Activity | 0 | ALA5155924 | NA | Homo sapiens | |||||
11. | ALA5191747 | 5cd | Activity | = | 80.56 | % | ALA5155924 | % | Homo sapiens | |||
12. | ALA5177960 | 5cc | Activity | = | 9.49 | % | ALA5155924 | % | Homo sapiens | |||
13. | ALA5178881 | 5cb | Activity | = | 96.73 | % | ALA5155924 | % | Homo sapiens | |||
14. | ALA5187212 | 5ca | Activity | 0 | ALA5155924 | NA | Homo sapiens | |||||
15. | ALA5187124 | (3S)5bf | Activity | = | 69.8 | % | ALA5155924 | % | Homo sapiens | |||
16. | ALA5197730 | (3R)5bf | Activity | = | 49.65 | % | ALA5155924 | % | Homo sapiens | |||
17. | ALA5175501 | (3S)5be | Activity | = | 62.37 | % | ALA5155924 | % | Homo sapiens | |||
18. | ALA5185166 | (3R)5be | Activity | = | 63.28 | % | ALA5155924 | % | Homo sapiens | |||
19. | ALA5197794 | 5bf | Activity | 0 | ALA5155924 | NA | Homo sapiens | |||||
20. | ALA5201636 | 5be | Activity | 0 | ALA5155924 | NA | Homo sapiens |