# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | AP-III-a4 (ENOblock) | 23 | IC50 | = | 0.576 | uM | ALA3386525 | 6.24 | nM | Homo sapiens | ||
2. | N-(4-{3-[2-(methylcarbamoyl)ethyl]-5-[4'-(trifluoromethyl)-[1,1'-biphenyl]-4-yl]-1H-pyrazol-1-yl}phenyl)prop-2-ynamide | 1; Tr-87 | Activity | 0 | ALA4415380 | Active | Homo sapiens | |||||
3. | ALA4643988 | VCY15 | IC50 | = | 7840 | nM | ALA4621999 | 5.11 | nM | Homo sapiens | ||
4. | TH-302 | 3b, TH-302 | IC50 | = | 897 | nM | ALA4621999 | 6.05 | nM | Homo sapiens | ||
5. | ALA4647008 | POMHEX | IC50 | = | 1814 | nM | ALA4621999 | 5.74 | nM | Homo sapiens | ||
6. | ALA4643988 | VCY15 | IC50 | = | 5764 | nM | ALA4621998 | 5.24 | nM | Homo sapiens | ||
7. | TH-302 | 3b, TH-302 | IC50 | = | 301 | nM | ALA4621998 | 6.52 | nM | Homo sapiens | ||
8. | ALA4647008 | POMHEX | IC50 | = | 2806 | nM | ALA4621998 | 5.55 | nM | Homo sapiens | ||
9. | ALA4643988 | VCY15 | IC50 | = | 21106 | nM | ALA4621996 | 4.68 | nM | Homo sapiens | ||
10. | TH-302 | 3b, TH-302 | IC50 | = | 4838 | nM | ALA4621996 | 5.32 | nM | Homo sapiens | ||
11. | ALA4647008 | POMHEX | IC50 | = | 2406 | nM | ALA4621996 | 5.62 | nM | Homo sapiens | ||
12. | ALA4643988 | VCY15 | IC50 | = | 25887 | nM | ALA4621995 | 4.59 | nM | Homo sapiens | ||
13. | TH-302 | 3b, TH-302 | IC50 | = | 2554 | nM | ALA4621995 | 5.59 | nM | Homo sapiens | ||
14. | ALA4647008 | POMHEX | IC50 | = | 720 | nM | ALA4621995 | 6.14 | nM | Homo sapiens | ||
15. | ALA4633981 | FLM37 | IC50 | = | 4020 | nM | ALA4621993 | 5.40 | nM | Homo sapiens | ||
16. | ALA4647008 | POMHEX | IC50 | = | 2148 | nM | ALA4621993 | 5.67 | nM | Homo sapiens | ||
17. | Hex | HEX | IC50 | > | 100000 | nM | ALA4621993 | nM | Homo sapiens | |||
18. | ALA4633981 | FLM37 | IC50 | = | 3945 | nM | ALA4621992 | 5.40 | nM | Homo sapiens | ||
19. | ALA4647008 | POMHEX | IC50 | = | 604 | nM | ALA4621992 | 6.22 | nM | Homo sapiens | ||
20. | Hex | HEX | IC50 | > | 100000 | nM | ALA4621992 | nM | Homo sapiens |